INHIBITION OF SPARTEINE OXIDATION IN HUMAN-LIVER BY TRICYCLIC ANTI-DEPRESSANTS AND OTHER DRUGS

被引:76
作者
OTTON, SV
INABA, T
KALOW, W
机构
关键词
D O I
10.1016/0024-3205(83)90315-6
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
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页码:795 / 800
页数:6
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共 20 条
[1]   PHARMACOGENETIC COVARIATION OF DEFECTIVE N-OXIDATION OF SPARTEINE AND 4-HYDROXYLATION OF DEBRISOQUINE [J].
BERTILSSON, L ;
DENGLER, HJ ;
EICHELBAUM, M ;
SCHULZ, HU .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 17 (02) :153-155
[2]  
COCCIA PF, 1967, J PHARMACOL EXP THER, V157, P446
[3]   INFLUENCE OF THE GENETICALLY CONTROLLED DEFICIENCY IN DEBRISOQUINE HYDROXYLATION ON ANTIPYRINE METABOLITE FORMATION [J].
DANHOF, M ;
IDLE, JR ;
TEUNISSEN, MWE ;
SLOAN, TP ;
BREIMER, DD ;
SMITH, RL .
PHARMACOLOGY, 1981, 22 (06) :349-358
[4]   APPARENT MICHAELIS CONSTANTS FOR METABOLISM OF (UREYL-C-14)TOLBUTAMIDE BY HUMAN LIVER MICROSOMAL PREPARATIONS [J].
DARBY, FJ ;
EVANS, DAP ;
GRUNDY, RK .
BIOCHEMICAL PHARMACOLOGY, 1972, 21 (03) :407-&
[5]  
Dixon M., 1964, ENZYMES, P328
[6]  
EICHELBAUM M, 1982, CLIN PHARMACOKINET, V7, P1, DOI 10.2165/00003088-198207010-00001
[7]  
EICHELBAUM M, 1975, THESIS U BONN
[8]  
IDLE JR, 1979, BRIT J PHARMACOL, V66, pP430
[9]   DEFICIENT METABOLISM OF DEBRISOQUINE AND SPARTEINE [J].
INABA, T ;
OTTON, SV ;
KALOW, W .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1980, 27 (04) :547-549
[10]   SPECTROPHOTOMETRIC AND TURBIDIMETRIC METHODS FOR MEASURING PROTEINS [J].
LAYNE, E .
METHODS IN ENZYMOLOGY, 1957, 3 :447-454