A METABOLITE OF BUSPIRONE INCREASES LOCUS COERULEUS ACTIVITY VIA ALPHA2-RECEPTOR BLOCKADE

被引:35
作者
ENGBERG, G
机构
关键词
D O I
10.1007/BF01578749
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:91 / 98
页数:8
相关论文
共 44 条
[1]   TOLERANCE OF LOCUS COERULEUS NEURONS TO MORPHINE AND SUPPRESSION OF WITHDRAWAL RESPONSE BY CLONIDINE [J].
AGHAJANIAN, GK .
NATURE, 1978, 276 (5684) :186-188
[2]   EVIDENCE FOR NOREPINEPHRINE-MEDIATED COLLATERAL INHIBITION OF LOCUS COERULEUS NEURONS [J].
AGHAJANIAN, GK ;
CEDARBAUM, JM ;
WANG, RY .
BRAIN RESEARCH, 1977, 136 (03) :570-577
[3]  
ASTONJONES G, 1981, J NEUROSCI, V1, P887
[4]  
ASTONJONES G, 1981, J NEUROSCI, V1, P879
[5]   DISPOSITION OF THE PSYCHOTROPIC-DRUGS BUSPIRONE, MJ-13805 AND PIRIBEDIL, AND OF THEIR COMMON ACTIVE METABOLITE 1-(2-PYRIMIDINYL)-PIPERAZINE IN THE RAT [J].
CACCIA, S ;
FONG, MH ;
GUISO, G .
XENOBIOTICA, 1985, 15 (10) :835-844
[6]   1-(2-PYRIMIDINYL)-PIPERAZINE AS ACTIVE METABOLITE OF BUSPIRONE IN MAN AND RAT [J].
CACCIA, S ;
CONTI, I ;
VIGANO, G ;
GARATTINI, S .
PHARMACOLOGY, 1986, 33 (01) :46-51
[7]   DISPOSITION AND METABOLISM OF BUSPIRONE AND ITS METABOLITE 1-(2-PYRIMIDINYL)-PIPERAZINE IN THE RAT [J].
CACCIA, S ;
MUGLIA, M ;
MANCINELLI, A ;
GARATTINI, S .
XENOBIOTICA, 1983, 13 (03) :147-153
[8]   ACTIVATION OF LOCUS COERULEUS NEURONS BY PERIPHERAL STIMULI - MODULATION BY A COLLATERAL INHIBITORY MECHANISM [J].
CEDARBAUM, JM ;
AGHAJANIAN, GK .
LIFE SCIENCES, 1978, 23 (13) :1383-1392
[9]   NORADRENERGIC NEURONS OF LOCUS COERULEUS - INHIBITION BY EPINEPHRINE AND ACTIVATION BY ALPHA-ANTAGONIST PIPEROXANE [J].
CEDARBAUM, JM ;
AGHAJANIAN, GK .
BRAIN RESEARCH, 1976, 112 (02) :413-419
[10]  
COLE JO, 1982, J CLIN PSYCHIAT, V43, P69