THERMODYNAMIC ASPECTS OF DRUG RECEPTOR INTERACTIONS

被引:47
作者
HITZEMANN, R [1 ]
机构
[1] VET ADM MED CTR, DIV PSYCHOBIOL, PSYCHIAT SERV, NORTHPORT, NY 11768 USA
关键词
D O I
10.1016/0165-6147(88)90068-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:408 / 411
页数:4
相关论文
共 31 条
  • [1] TEMPERATURE COEFFICIENTS OF AFFINITY CONSTANTS FOR THE BINDING OF ANTAGONISTS TO MUSCARINIC RECEPTORS IN THE RAT CEREBRAL-CORTEX
    BARLOW, RB
    BIRDSALL, NJM
    HULME, EC
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1979, 66 (04) : 587 - 590
  • [2] THE BINDING OF AGONISTS AND ANTAGONISTS TO RAT LUNG BETA-ADRENERGIC RECEPTORS AS INVESTIGATED BY THERMODYNAMICS AND STRUCTURE-ACTIVITY-RELATIONSHIPS
    BREE, F
    ELTAYAR, N
    VANDEWATERBEEMD, H
    TESTA, B
    TILLEMENT, JP
    [J]. JOURNAL OF RECEPTOR RESEARCH, 1986, 6 (5-6): : 381 - 409
  • [3] CHANG KJ, 1981, MOL PHARMACOL, V20, P1
  • [4] Cho T M, 1979, Adv Biochem Psychopharmacol, V20, P69
  • [5] CONTRERAS ML, 1986, J PHARMACOL EXP THER, V237, P165
  • [6] Cornish-Bowden A, 1976, PRINCIPLES ENZYME KI
  • [7] DISCRIMINATION BY TEMPERATURE OF OPIATE AGONIST AND ANTAGONIST RECEPTOR-BINDING
    CREESE, I
    PASTERNAK, GW
    PERT, CB
    SNYDER, SH
    [J]. LIFE SCIENCES, 1975, 16 (12) : 1837 - 1842
  • [8] CREESE I, 1987, PSYCHOPHARMACOLOGY 3, P257
  • [9] Edelhoch H, 1976, Adv Protein Chem, V30, P183, DOI 10.1016/S0065-3233(08)60480-5
  • [10] BINDING-ENERGY AND THE ACTIVATION OF HORMONE RECEPTORS
    FRANKLIN, TJ
    [J]. BIOCHEMICAL PHARMACOLOGY, 1980, 29 (06) : 853 - 856