BARBITURATES ALLOSTERICALLY INHIBIT GABA ANTAGONIST AND BENZODIAZEPINE INVERSE AGONIST BINDING

被引:38
作者
WONG, EHF
SNOWMAN, AM
LEEBLUNDBERG, LMF
OLSEN, RW
机构
[1] UNIV CALIF LOS ANGELES,SCH MED,DEPT PHARMACOL,LOS ANGELES,CA 90024
[2] UNIV CALIF RIVERSIDE,DIV BIOMED SCI,RIVERSIDE,CA 92521
[3] UNIV CALIF RIVERSIDE,DEPT BIOCHEM,RIVERSIDE,CA 92521
关键词
D O I
10.1016/0014-2999(84)90252-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:205 / 212
页数:8
相关论文
共 39 条
  • [1] CHLORIDE-DEPENDENT STIMULATION OF GABA AND BENZODIAZEPINE RECEPTOR-BINDING BY PENTOBARBITAL
    ASANO, T
    OGASAWARA, N
    [J]. BRAIN RESEARCH, 1981, 225 (01) : 212 - 216
  • [2] ETOMIDATE STEREOSPECIFICALLY STIMULATES FOREBRAIN, BUT NOT CEREBELLAR, DIAZEPAM-H-3 BINDING
    ASHTON, D
    GEERTS, R
    WATERKEYN, C
    LEYSEN, JE
    [J]. LIFE SCIENCES, 1981, 29 (25) : 2631 - 2636
  • [3] GABA REDUCES BINDING OF H-3-LABELED METHYL BETA-CARBOLINE-3-CARBOXYLATE TO BRAIN BENZODIAZEPINE RECEPTORS
    BRAESTRUP, C
    NIELSEN, M
    [J]. NATURE, 1981, 294 (5840) : 472 - 474
  • [4] BROWNER M, 1981, J NEUROSCI, V1, P514
  • [5] MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES
    COSTA, E
    GUIDOTTI, A
    [J]. ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 : 531 - 545
  • [6] IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL
    COSTA, T
    RODBARD, D
    PERT, CB
    [J]. NATURE, 1979, 277 (5694) : 315 - 317
  • [7] ANIONIC PERMEABILITY OF INHIBITORY POSTSYNAPTIC MEMBRANE OF HIPPOCAMPAL PYRAMIDAL CELLS
    ECCLES, J
    NICOLL, RA
    OSHIMA, T
    RUBIA, FJ
    [J]. PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1977, 198 (1133): : 345 - 361
  • [8] AN ALLOSTERIC MODEL FOR BENZODIAZEPINE RECEPTOR FUNCTION
    EHLERT, FJ
    ROESKE, WR
    GEE, KW
    YAMAMURA, HI
    [J]. BIOCHEMICAL PHARMACOLOGY, 1983, 32 (16) : 2375 - 2383
  • [9] ENNA SJ, 1977, MOL PHARMACOL, V13, P442
  • [10] GAMMA-AMINOBUTYRIC ACID AND BENZODIAZEPINE RECEPTORS - COPURIFICATION AND CHARACTERIZATION
    GAVISH, M
    SNYDER, SH
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (03): : 1939 - 1942