SPIRO-[4H-PYRROLO[1,2-A][1,4]BENZODIAZEPINE-4,4'-PIPERIDINE] DERIVATIVES AS POTENTIAL NOOTROPIC AGENTS - A SIMPLE ONE-POT SYNTHESIS

被引：10

作者：

MASSA, S ^{[1
]}

MAI, A ^{[1
]}

ARTICO, M ^{[1
]}

机构：

[1] UNIV ROME LA SAPIENZA,DIPARTIMENTO STUDI FARMACEUT,P LE ALDO MORO 5,I-00185 ROME,ITALY

来源：

SYNTHETIC COMMUNICATIONS | 1990年 / 20卷 / 22期

关键词：

D O I：

10.1080/00397919008051597

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Some derivatives of a new heterocyclic ring, spiro-[4H-pyrrolo[1,2a][1,4]benzodiazepine-4,4'-piperidine], have been obtained in very good yields by a simple one-pot reaction using 1-(2-aminomethylphenyl)-1H-pyrrole and 1-substituted 4-oxopiperidines as the synthones.

引用

页码：3537 / 3545

页数：9

共 6 条

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[3] SYNTHESIS OF 5,6-DIHYDRO-4H-PYRROLO[1,2-A] [1,4]BENZODIAZEPINES [J].

CHEESEMAN, GWH ;

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[4]

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[5]

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[6]

MATTSON RJ, 1988, ANNU REP MED CHEM, V23, P29

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