MOLECULAR AND STRUCTURAL BASIS OF RESTING AND USE-DEPENDENT BLOCK OF SODIUM CURRENT DEFINED USING DISOPYRAMIDE ANALOGS

被引:41
作者
YEH, JZ
TENEICK, RE
机构
关键词
D O I
10.1016/S0006-3495(87)83317-9
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
引用
收藏
页码:123 / 135
页数:13
相关论文
共 28 条
[1]   DESTRUCTION OF SODIUM CONDUCTANCE INACTIVATION IN SQUID AXONS PERFUSED WITH PRONASE [J].
ARMSTRONG, CM ;
BEZANILLA, F ;
ROJAS, E .
JOURNAL OF GENERAL PHYSIOLOGY, 1973, 62 (04) :375-391
[2]   REPLACEMENT OF PROTOPLASM OF A GIANT NERVE FIBRE WITH ARTIFICIAL SOLUTIONS [J].
BAKER, PF ;
SHAW, TI ;
HODGKIN, AL .
NATURE, 1961, 190 (477) :885-+
[3]  
BOKESCH PM, 1986, J PHARMACOL EXP THER, V237, P773
[4]   INTERACTIONS BETWEEN QUATERNARY LIDOCAINE, THE SODIUM-CHANNEL GATES, AND TETRODOTOXIN [J].
CAHALAN, MD ;
ALMERS, W .
BIOPHYSICAL JOURNAL, 1979, 27 (01) :39-55
[5]   BLOCK OF SODIUM CONDUCTANCE AND GATING CURRENT IN SQUID GIANT-AXONS POISONED WITH QUATERNARY STRYCHNINE [J].
CAHALAN, MD ;
ALMERS, W .
BIOPHYSICAL JOURNAL, 1979, 27 (01) :57-73
[6]   LOCAL-ANESTHETIC BLOCK OF SODIUM CHANNELS IN NORMAL AND PRONASE-TREATED SQUID GIANT-AXONS [J].
CAHALAN, MD .
BIOPHYSICAL JOURNAL, 1978, 23 (02) :285-311
[7]  
CAHALAN MD, 1976, BIOPHYS J, V16, pA76
[8]   IMPORTANCE OF PHYSICOCHEMICAL PROPERTIES IN DETERMINING THE KINETICS OF THE EFFECTS OF CLASS-I ANTI-ARRHYTHMIC DRUGS ON MAXIMUM RATE OF DEPOLARIZATION IN GUINEA-PIG VENTRICLE [J].
CAMPBELL, TJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 80 (01) :33-40
[9]  
COURTNEY KR, 1975, J PHARMACOL EXP THER, V195, P225
[10]  
COURTNEY KR, 1980, J PHARMACOL EXP THER, V213, P114