CORRELATIONS AMONG MINIMAL NEUROTOXICITY, ANTI-CONVULSANT ACTIVITY, AND DISPLACING POTENCIES IN [FLUNITRAZEPAM-H-3 BINDING OF BENZODIAZEPINES

被引:20
作者
CHWEH, AY
SWINYARD, EA
WOLF, HH
KUPFERBERG, HJ
机构
[1] UNIV UTAH,COLL PHARM,DEPT BIOCHEM PHARMACOL & TOXICOL,SALT LAKE CITY,UT 84112
[2] NINCDS,EPILEPSY BRANCH,NEUROL DISORDERS BRANCH,BETHESDA,MD 20205
关键词
D O I
10.1111/j.1528-1157.1983.tb04629.x
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:668 / 677
页数:10
相关论文
共 24 条
[1]   STRYCHNINE AS A POTENT INHIBITOR OF THE BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M .
BRAIN RESEARCH BULLETIN, 1980, 5 :681-684
[2]   SPECIFIC BENZODIAZEPINE RECEPTORS IN RAT-BRAIN CHARACTERIZED BY HIGH-AFFINITY [DIAZEPAM-H-3] BINDING - (AFFINITY BINDING DIAZEPAM ANXIOLYTIC ACTIVITY BRAIN MEMBRANES REGIONAL DISTRIBUTION) [J].
BRAESTRUP, C ;
SQUIRES, RF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (09) :3805-3809
[3]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[4]   BENZODIAZEPINES AND CENTRAL GLYCINE RECEPTORS [J].
CURTIS, DR ;
GAME, CJA ;
LODGE, D .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 56 (03) :307-311
[5]  
ENNA SJ, 1977, MOL PHARMACOL, V13, P442
[6]   EFFECT OF PICROTOXIN ON BENZODIAZEPINE RECEPTORS AND GABA RECEPTORS WITH REFERENCE TO THE EFFECT OF CL- ION [J].
FUJIMOTO, M ;
OKABAYASHI, T .
LIFE SCIENCES, 1981, 28 (08) :895-901
[7]  
Haefely W, 1975, Adv Biochem Psychopharmacol, P131
[8]   MODULATION BY PICROTOXIN AND IPTBO OF FLUNITRAZEPAM-H-3 BINDING TO THE GABA-BENZODIAZEPINE RECEPTOR COMPLEX OF RAT CEREBELLUM [J].
KAROBATH, M ;
DREXLER, G ;
SUPAVILAI, P .
LIFE SCIENCES, 1981, 28 (03) :307-313
[9]   ANTIEPILEPTIC DRUG DEVELOPMENT .2. ANTICONVULSANT DRUG SCREENING [J].
KRALL, RL ;
PENRY, JK ;
WHITE, BG ;
KUPFERBERG, HJ ;
SWINYARD, EA .
EPILEPSIA, 1978, 19 (04) :409-428
[10]  
Lippa A., 1979, ANXIOLYTICS, P41