SERUM CONCENTRATIONS AND URINARY-EXCRETION OF PINACIDIL AND ITS MAJOR METABOLITE, PINACIDIL PYRIDINE-N-OXIDE FOLLOWING IV AND ORAL-ADMINISTRATION IN HEALTHY-VOLUNTEERS

被引:17
作者
MCBURNEY, A
FARROW, PR
AINSWORTH, S
WARD, JW
机构
关键词
D O I
10.1111/j.1365-2125.1985.tb02618.x
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:91 / 94
页数:4
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共 9 条
[1]   N''-CYANO-N-4-PYRIDYL-N'-1,2,2-TRIMETHYLPROPYLGUANIDINE, MONOHYDRATE (P 1134) - A NEW, POTENT VASODILATOR [J].
ARRIGONIMARTELLI, E ;
NIELSEN, CK ;
OLSEN, UB ;
PETERSEN, HJ .
EXPERIENTIA, 1980, 36 (04) :445-447
[2]  
CARLSEN JE, 1981, CLIN PHYSL, V1, P357
[3]   METABOLISM OF THE NEW ANTIHYPERTENSIVE AGENT PINACIDIL IN RAT, DOG AND MAN [J].
EILERTSEN, E ;
MAGNUSSEN, MP ;
PETERSEN, HJ ;
RASTRUPANDERSEN, N ;
SORENSEN, H ;
ARRIGONIMARTELLI, E .
XENOBIOTICA, 1982, 12 (03) :187-196
[4]   PHARMACOKINETICS AND DISTRIBUTION OF THE NEW ANTIHYPERTENSIVE AGENT PINACIDIL IN RAT, DOG AND MAN [J].
EILERTSEN, E ;
HART, JW ;
MAGNUSSEN, MP ;
SORENSEN, H ;
ARRIGONIMARTELLI, E .
XENOBIOTICA, 1982, 12 (03) :177-185
[5]  
FARROW PR, 1984, EUR J CLIN PHARM
[6]  
MUIESAN G, 1983, CLIN PHARMACOL THER, V33, P229
[7]   SYNTHESIS AND HYPOTENSIVE ACTIVITY OF N-ALKYL-N'-CYANO-N'-PYRIDYLGUANIDINES [J].
PETERSEN, HJ ;
NIELSEN, CK ;
ARRIGONIMARTELLI, E .
JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (08) :773-781
[8]   HEMODYNAMIC CHARACTERIZATION OF PINACIDIL IN RATS - COMPARISON WITH HYDRALAZINE [J].
THOOLEN, MJMC ;
VANMEEL, JCA ;
WILFFERT, B ;
TIMMERMANS, PBMWM ;
VANZWIETEN, PA .
PHARMACOLOGY, 1983, 27 (05) :245-254
[9]   PHARMACOKINETICS AND HYPOTENSIVE EFFECT IN HEALTHY-VOLUNTEERS OF PINACIDIL, A NEW POTENT VASODILATOR [J].
WARD, JW ;
MCBURNEY, A ;
FARROW, PR ;
SHARP, P .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 26 (05) :603-608