ASYMMETRIC-SYNTHESIS OF THE ENKEPHALINASE INHIBITOR THIORPHAN

被引：121

作者：

EVANS, DA ^{[1
]}

MATHRE, DJ ^{[1
]}

SCOTT, WL ^{[1
]}

机构：

[1] ELI LILLY RES LABS, INDIANAPOLIS, IN 46206 USA

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1985年 / 50卷 / 11期

关键词：

D O I：

10.1021/jo00211a008

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1830 / 1835

页数：6

共 37 条

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[3] INHIBITION OF ENKEPHALIN METABOLISM BY, AND ANTI-NOCICEPTIVE ACTIVITY OF, BESTATIN, AN AMINOPEPTIDASE INHIBITOR
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[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 83 (3-4) : 283 - 288
[5] POTENTIATION OF STRESS-INDUCED ANALGESIA (SIA) BY THIORPHAN AND ITS BLOCK BY NALOXONE
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[6] ALPHA-METHOXY-ALPHA-TRIFLUOROMETHYLPHENYLACETIC ACID, A VERSATILE REAGENT FOR DETERMINATION OF ENANTIOMERIC COMPOSITION OF ALCOHOLS AND AMINES
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[7] 2-OXAZOLIDONES
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[8] Evans D. A., 1982, ALDRICHIM ACTA, V15, P23
[9] NEW ASYMMETRIC DIELS-ALDER CYCLOADDITION REACTIONS - CHIRAL ALPHA,BETA-UNSATURATED CARBOXIMIDES AS PRACTICAL CHIRAL ACRYLATE AND CROTONATE DIENOPHILE SYNTHONS
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[10] ENANTIOSELECTIVE ALDOL CONDENSATIONS .2. ERYTHRO-SELECTIVE CHIRAL ALOL CONDENSATIONS VIA BORON ENOLATES
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