SYNTHESIS AND EVALUATION OF FLUORINATED DERIVATIVES OF FENTANYL AS CANDIDATES FOR OPIATE RECEPTOR STUDIES USING POSITRON EMISSION TOMOGRAPHY

被引：22

作者：

HWANG, DR

FELIU, AL

WOLF, AP

MACGREGOR, RR

FOWLER, JS

ARNETT, CD

HOLLAND, MJ

CARR, K

SIMON, EJ

机构：

[1] BROOKHAVEN NATL LAB,DEPT CHEM,UPTON,NY 11973

[2] NYU MED CTR,DEPT PSYCHIAT,NEW YORK,NY 10016

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 1986年 / 23卷 / 03期

关键词：

D O I：

10.1002/jlcr.2580230306

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：277 / 293

页数：17

共 31 条

[1] [F-18] N-METHYLSPIROPERIDOL - THE RADIOLIGAND OF CHOICE FOR PETT STUDIES OF THE DOPAMINE RECEPTOR IN HUMAN-BRAIN [J].

ARNETT, CD ;

FOWLER, JS ;

WOLF, AP ;

SHIUE, CY ;

MCPHERSON, DW .

LIFE SCIENCES, 1985, 36 (14) :1359-1366

[2] COMPARISON OF 3 F-18-LABELED BUTYROPHENONE NEUROLEPTIC DRUGS IN THE BABOON USING POSITRON EMISSION TOMOGRAPHY [J].

ARNETT, CD ;

SHIUE, CY ;

WOLF, AP ;

FOWLER, JS ;

LOGAN, J ;

WATANABE, M .

JOURNAL OF NEUROCHEMISTRY, 1985, 44 (03) :835-844

[3] DISPLACEMENT OF A NITRO-GROUP BY [F-18]-LABELED FLUORIDE-ION - A NEW ROUTE TO ARYL FLUORIDES OF HIGH SPECIFIC ACTIVITY [J].

ATTINA, M ;

CACACE, F ;

WOLF, AP .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1983, (03) :108-109

[4] LABELED ARYL FLUORIDES FROM THE NUCLEOPHILIC DISPLACEMENT OF ACTIVATED NITRO-GROUPS BY F-18-F- [J].

ATTINA, M ;

CACACE, F ;

WOLF, AP .

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1983, 20 (04) :501-514

[5] HALIDE CATALYSIS IN BROMINATION OF DEOXYBENZOIN [J].

CIECIUCH, RF ;

WESTHEIMER, FH .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1963, 85 (17) :2591-&

[6]

DANNALS RF, 1985, INT J APPL RADIAT IS, V36, P303, DOI 10.1016/0020-708X(85)90089-4

[7]

DANNALS RF, 1982, J LABELLED COMPD RAD, V19, P1493

[8]

FROST JJ, 1985, J COMPUT ASSIST TOMO, V9, P231, DOI 10.1097/00004728-198503000-00001

[9]

FROST JJ, 1984, ANN NEUROL, V15, pS85

[10] REDUCTION OF ALDEHYDES AND KETONES TO ALCOHOLS AND HYDROCARBONS THROUGH USE OF ORGANOSILANE-BORON TRIFLUORIDE SYSTEM [J].

FRY, JL ;

ORFANOPOULOS, M ;

ADLINGTON, MG ;

DITTMAN, WR ;

SILVERMAN, SB .

JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (02) :374-375

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