CONCISE GENERAL-SYNTHESIS OF ALPHA,GAMMA-DISUBSTITUTED BETA-AMINO KETONES FROM BETA-LACTAMS

被引：37

作者：

PALOMO, C

AIZPURUA, JM

GARCIA, JM

ITURBURU, M

ODRIOZOLA, JM

机构：

[1] Departamento de Química Orgánica, Facultad de Química, Universidad del Pais Vasco, Apdo 1072

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1994年 / 59卷 / 18期

关键词：

D O I：

10.1021/jo00097a020

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

alpha,gamma-Disubstituted beta-amino ketones were obtained by ring opening of 3,4-disubstituted N-Boc-beta-lactams, promoted by Grignard and organocuprate reagents.

引用

页码：5184 / 5188

页数：5

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