SYNTHESIS OF 5-FLUORO-1,3-DIOXIN-4-ONES - VERSATILE BUILDING-BLOCKS OF FLUORINATED COMPOUNDS

被引：18

作者：

SATO, M

KANEKO, C

IWAOKA, T

KOBAYASHI, Y

IIDA, T

机构：

[1] TOHOKU UNIV,INST PHARMACEUT,SENDAI,MIYAGI 980,JAPAN

[2] CHUGAI PHARMACEUT CO LTD,PROD TECHNOL RES LAB,KITA KU,TOKYO 115,JAPAN

[3] TOKYO COLL PHARM,HACHIOJI,TOKYO 19203,JAPAN

[4] DAIKIN IND LTD,MEC LAB,TSUKUBA,IBARAKI 305,JAPAN

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1991年 / 10期

关键词：

D O I：

10.1039/c39910000699

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Fluorination of 5,6-unsubstituted 1,3-dioxin-4-ones by fluorine followed by treatment with triethylamine affords the title compounds, which can be converted into fluorinated derivatives of either formylacetic acid or of heterocyclic systems.

引用

页码：699 / 700

页数：2

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