ANTIMALARIALS .14. 5-(ARYLOXY)-4-METHYLPRIMAQUINE ANALOGS - A HIGHLY EFFECTIVE SERIES OF BLOOD AND TISSUE SCHIZONTICIDAL AGENTS

被引：52

作者：

LAMONTAGNE, MP ^{[1
]}

BLUMBERGS, P ^{[1
]}

STRUBE, RE ^{[1
]}

机构：

[1] WALTER REED ARMY INST RES,WASHINGTON,DC 20012

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1982年 / 25卷 / 09期

关键词：

D O I：

10.1021/jm00351a017

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1094 / 1097

页数：4

共 10 条

[1] MODIFICATIONS OF PRIMAQUINE AS ANTIMALARIALS .1. 5-PHENOXY DERIVATIVES OF PRIMAQUINE [J].

CHEN, EH ;

SAGGIOMO, AJ ;

TANABE, K ;

VERMA, BL ;

NODIFF, EA .

JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (08) :1107-1109

[2] EVALUATING NEW ANTIMALARIAL-DRUGS AGAINST TROPHOZOITE INDUCED PLASMODIUM-CYNOMOLGI MALARIA IN RHESUS-MONKEYS [J].

DAVIDSON, DE ;

JOHNSEN, DO ;

TANTICHAROENYOS, P ;

HICKMAN, RL ;

KINNAMON, KE .

AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1976, 25 (01) :26-33

[3] SYNTHESIS OF PRIMAQUINE AND CERTAIN OF ITS ANALOGS [J].

ELDERFIELD, RC ;

MERTEL, HE ;

MITCH, RT ;

WEMPEN, IM ;

WERBLE, E .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1955, 77 (18) :4816-4819

[4] THE SYNTHESIS OF 5-HYDROXY-8-NITROQUINOLINE AND CERTAIN OF ITS DERIVATIVES [J].

FUSON, RC ;

BAUMAN, RA ;

HOWARD, E ;

MARVELL, EN .

JOURNAL OF ORGANIC CHEMISTRY, 1947, 12 (06) :799-806

[5] ANTIMALARIALS .6. SYNTHESIS, ANTIMALARIAL ACTIVITY, AND CONFIGURATIONS OF RACEMIC ALPHA-(2-PIPERIDYL)-4-PYRIDINEMETHANOLS [J].

LAMONTAG.MP ;

MARKOVAC, A ;

BLUMBERG.P .

JOURNAL OF MEDICINAL CHEMISTRY, 1974, 17 (05) :519-523

[6] ANTIMALARIALS .13. 5-ALKOXY ANALOGS OF 4-METHYLPRIMAQUINE [J].

LAMONTAGNE, MP ;

MARKOVAC, A ;

KHAN, MS .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (08) :964-968

[7] ANTIMALARIALS .10. SYNTHESIS OF 4-SUBSTITUTED PRIMAQUINE ANALOGS AS CANDIDATE ANTIMALARIALS [J].

LAMONTAGNE, MP ;

MARKOVAC, A ;

MENKE, JR .

JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (09) :1122-1127

[8] ANTIMALARIAL PHENANTHRENE AMINO ALCOHOLS .2. TRIFLUOROMETHYL-CONTAINING 9-PHENANTHRENEMETHANOLS [J].

NODIFF, EA ;

OTOMASU, H ;

VERMA, BL ;

TYAGI, MP ;

SHINBO, M ;

SAGGIOMO, AJ ;

TANABE, K ;

CHEN, EH ;

MATSUURA, S ;

MOROSAWA, S ;

KIKUCHI, T ;

KONDO, Y .

JOURNAL OF MEDICINAL CHEMISTRY, 1972, 15 (07) :775-&

[9] 2,4,7-TRIAMINO-6-ORTHO-SUBSTITUTED ARYLPTERIDINES . A NEW SERIES OF POTENT ANTIMALARIAL AGENTS [J].

OSDENE, TS ;

RUSSELL, PB ;

RANE, L .

JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (03) :431-&

[10] ACTIVITY OF A REPOSITORY FORM OF 4,6-DIAMINO-1-(P-CHLOROPHENYL)-1,2-DIHYDRO-2,2-DIMETHYL-S-TRIAZINE AGAINST INFECTIONS WITH PLASMODIUM CYNOMOLGI [J].

SCHMIDT, LH ;

FISHER, KF ;

ROSSAN, RN .

AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1963, 12 (04) :494-&

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