THE CONTRIBUTION OF INTRINSIC ACTIVITY TO THE ACTION OF OPIOIDS INVITRO

被引:121
作者
MILLER, L
SHAW, JS
WHITING, EM
机构
关键词
D O I
10.1111/j.1476-5381.1986.tb10202.x
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:595 / 601
页数:7
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共 19 条
[1]  
ARIENS EJ, 1964, MOL PHARMACOL, P394
[2]   MU-RECEPTOR BINDING IN PHYSIOLOGICAL MEDIA - COMPARISON WITH ISOLATED TISSUE DATA [J].
CARROLL, JA ;
MILLER, L ;
SHAW, JS ;
DOWNES, CP .
NEUROPEPTIDES, 1984, 5 (1-3) :89-92
[3]  
HENDERSON G, 1982, BR J PHARM S, V75, pP29
[4]   ASSESSMENT IN GUINEA-PIG ILEUM AND MOUSE VAS-DEFERENS OF BENZOMORPHANS WHICH HAVE STRONG ANTINOCICEPTIVE ACTIVITY BUT DO NOT SUBSTITUTE FOR MORPHINE IN DEPENDENT MONKEY [J].
HUTCHINSON, M ;
KOSTERLITZ, HW ;
LESLIE, FM ;
WATERFIELD, AA ;
TERENIUS, L .
BRITISH JOURNAL OF PHARMACOLOGY, 1975, 55 (04) :541-546
[5]   EVIDENCE FOR A SINGLE OPIOID RECEPTOR TYPE ON THE FIELD STIMULATED RAT VAS-DEFERENS [J].
LIAO, CS ;
DAY, AR ;
FREER, RJ .
LIFE SCIENCES, 1981, 29 (25) :2617-2622
[6]   ENDOGENOUS OPIOID PEPTIDES - MULTIPLE AGONISTS AND RECEPTORS [J].
LORD, JAH ;
WATERFIELD, AA ;
HUGHES, J ;
KOSTERLITZ, HW .
NATURE, 1977, 267 (5611) :495-499
[7]  
LORD JAH, 1976, OPIATES ENDOGENOUS O, P275
[9]  
MCKNIGHT AT, 1984, NEUROPEPTIDES, V5, P97, DOI 10.1016/0143-4179(84)90036-2
[10]   INCREASE IN POTENCIES OF OPIOID-PEPTIDES AFTER PEPTIDASE INHIBITION [J].
MCKNIGHT, AT ;
CORBETT, AD ;
KOSTERLITZ, HW .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 86 (3-4) :393-402