AN ALTERNATIVE APPROACH TO DEVELOPING DOPAMINE-RECEPTOR AGONISTS WITH CENTRAL PRE-SYNAPTIC ACTIONS FOLLOWING ORAL-ADMINISTRATION - A COMPARISON BETWEEN APOMORPHINE, BROMOCRIPTINE, AND THE NOVEL COMPOUND RDS-127 (2-DI-N-PROPYLAMINO-4,7-DIMETHOXYINDANE)

被引:8
作者
ARNERIC, SP [1 ]
LONG, JP [1 ]
机构
[1] UNIV IOWA, COLL MED, DEPT PHARMACOL, IOWA CITY, IA 52242 USA
关键词
D O I
10.1002/ddr.430030304
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:221 / 231
页数:11
相关论文
共 40 条
[31]  
SMITH RV, 1979, RES COMMUN CHEM PATH, V24, P483
[32]   CORRELATION OF BEHAVIORAL INHIBITION OR EXCITATION PRODUCED BY BROMOCRIPTINE WITH CHANGES IN BRAIN CATECHOLAMINE TURNOVER [J].
SNIDER, SR ;
HUTT, C ;
STEIN, B ;
PRASAD, ALN ;
FAHN, S .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1976, 28 (07) :563-566
[33]  
Steel R.G.D., 1960, PRINCIPLES PROCEDURE, P106
[34]   ANTAGONISM BY HALOPERIDOL OF LOCOMOTOR DEPRESSION INDUCED BY SMALL DOSES OF APOMORPHINE [J].
STROMBOM, U .
JOURNAL OF NEURAL TRANSMISSION, 1977, 40 (03) :191-194
[35]   INVOLVEMENT OF BOTH DOPAMINERGIC AND ALPHA-ADRENERGIC RECEPTORS IN THE HYPOMOTILITY INDUCED BY DIBENZOYL-6,7-ADTN [J].
SUMNERS, C ;
DEVRIES, JB ;
DIJKSTRA, D ;
HORN, AS .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (04) :541-550
[36]   SCHIZOPHRENIC SYMPTOMS IMPROVE WITH APOMORPHINE [J].
TAMMINGA, CA ;
SCHAFFER, MH ;
SMITH, RC ;
DAVIS, JM .
SCIENCE, 1978, 200 (4341) :567-569
[37]   TREATMENT OF SCHIZOPHRENIA WITH ERGOT DERIVATIVES [J].
TAMMINGA, CA ;
SCHAFFER, MH .
PSYCHOPHARMACOLOGY, 1979, 66 (03) :239-242
[38]  
TITELER M, 1979, COMMUN PSYCHOPHARMAC, V3, P411
[39]  
Trabucchi M, 1977, Adv Biochem Psychopharmacol, V16, P661
[40]   DOPAMINERGIC-NEURONS - INVIVO SYSTEM FOR MEASURING DRUG INTERACTIONS WITH PRESYNAPTIC RECEPTORS [J].
WALTERS, JR ;
ROTH, RH .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1976, 296 (01) :5-14