2-TRIFLUOROMETHYL AMINO-ACIDS .12. PEPTIDE MODIFICATION BY INTRODUCTION OF ALPHA-TRIFLUOROMETHYL ALPHA-AMINO-ACIDS VIA 4-TRIFLUOROMETHYL-1,3-OXAZOLIDIN-2,5-DIONES

被引：32

作者：

SCHIERLINGER, C ^{[1
]}

BURGER, K ^{[1
]}

机构：

[1] TECH UNIV MUNICH,INST ORGAN CHEM,LICHTENBERGSTR 4,W-8046 GARCHING,GERMANY

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 02期

关键词：

ALPHA-TRIFLUOROMETHYL ALPHA-AMINO ACIDS; LEUCHS ANHYDRIDES; PEPTIDE MODIFICATION;

D O I：

10.1016/0040-4039(92)88047-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Alpha-Trifluoromethyl substituted alpha-amino acids can be introduced into the N-terminal position of peptides on carboxyl group activation via Leuchs anhydrides.

引用

页码：193 / 194

页数：2

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