A FACILE PREPARATION OF 2-(2-ARYLETHYL)INDOLES AND 2-(AMINOMETHYL)INDOLES

被引：8

作者：

NAGARATHNAM, D

机构：

[1] Department of Medicinal Chemistry and Pharmacognosy, University of Illinois at Chicago, Chicago, Illinois, 60680

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1992年 / 29卷 / 06期

关键词：

D O I：

10.1002/jhet.5570290601

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An important process for the acid catalyzed cleavage of the benzoyl group from 3-benzoylindoles in high yield is identified and its application for the facile syntheses of 2-substituted indoles is demonstrated by preparing some 2-(2-arylethyl)- and 2-(aminomethyl)indoles from 1,3-dibenzoyl-2-bromomethylindole (7).

引用

页码：1371 / 1373

页数：3

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