SYNTHESIS AND RECEPTOR AFFINITIES OF SOME CONFORMATIONALLY RESTRICTED ANALOGS OF THE DOPAMINE D1 SELECTIVE LIGAND (5R)-8-CHLORO-2,3,4,5-TETRAHYDRO-3-METHYL-5-PHENYL-1H-3-BENZAZEPIN-7-OL

被引：79

作者：

BERGER, JG ^{[1
]}

CHANG, WK ^{[1
]}

CLADER, JW ^{[1
]}

HOU, D ^{[1
]}

CHIPKIN, RE ^{[1
]}

MCPHAIL, AT ^{[1
]}

机构：

[1] DUKE UNIV,PAUL M GROSS CHEM LAB,DEPT CHEM,DURHAM,NC 27706

来源：

关键词：

D O I：

10.1021/jm00128a038

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1913 / 1921

页数：9

共 16 条

[1] [Anonymous], 1974, INT TABLES XRAY CRYS, VIV
[2] BARNETT A, 1986, Drugs of the Future, V11, P49
[3] CHARACTERIZATION OF THE BINDING OF H-3-SCH 23390, A SELECTIVE D-1 RECEPTOR ANTAGONIST LIGAND, IN RAT STRIATUM
BILLARD, W
RUPERTO, V
CROSBY, G
IORIO, LC
BARNETT, A
[J]. LIFE SCIENCES, 1984, 35 (18) : 1885 - 1893
[4] CHIPKIN RE, 1988, J PHARMACOL EXP THER, V247, P1093
[5] SYNTHESIS, RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND ENANTIOSELECTIVITY OF 3',4'-DIHYDROXYNOMIFENSINE
DANDRIDGE, PA
KAISER, C
BRENNER, M
GAITANOPOULOS, D
DAVIS, LD
WEBB, RL
FOLEY, JJ
SARAU, HM
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (01) : 28 - 35
[6] Goldberg L I, 1977, Adv Biochem Psychopharmacol, V16, P251
[7] SIGNIFICANCE TESTS ON CRYSTALLOGRAPHIC R FACTOR
HAMILTON, WC
[J]. ACTA CRYSTALLOGRAPHICA, 1965, 18 : 502 - &
[8] SCH-23390 - THE 1ST SELECTIVE DOPAMINE D-1 ANTAGONIST
HYTTEL, J
[J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 91 (01) : 153 - 154
[9] Iorio L C, 1986, Adv Exp Med Biol, V204, P1
[10] IORIO LC, 1983, J PHARMACOL EXP THER, V226, P462