ORAL MORPHINE IN CANCER-PATIENTS - INVIVO KINETICS AND INVITRO HEPATIC GLUCURONIDATION

被引:134
作者
SAWE, J
KAGER, L
ENG, JOS
RANE, A
机构
[1] HUDDINGE HOSP, KAROLINSKA INST, DEPT CLIN PHARMACOL, S-14186 HUDDINGE, SWEDEN
[2] HUDDINGE HOSP, KAROLINSKA INST, DEPT SURG, S-14186 HUDDINGE, SWEDEN
关键词
D O I
10.1111/j.1365-2125.1985.tb02675.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:495 / 501
页数:7
相关论文
共 21 条
[1]  
AGENAS I, 1982, LAKRTIDNINGEN, V78, P287
[2]   THE GUT WALL METABOLISM OF ETHINYLESTRADIOL AND ITS CONTRIBUTION TO THE PRE-SYSTEMIC METABOLISM OF ETHINYLESTRADIOL IN HUMANS [J].
BACK, DJ ;
BRECKENRIDGE, AM ;
MACIVER, M ;
ORME, M ;
PURBA, HS ;
ROWE, PH ;
TAYLOR, I .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 13 (03) :325-330
[3]   DETERMINATION OF MICROSOMAL UDP-GLUCURONYLTRANSFERASE IN NEEDLE-BIOPSY SPECIMENS OF HUMAN LIVER [J].
BOCK, KW ;
BRUNNER, G ;
HOENSCH, H ;
HUBER, E ;
JOSTING, D .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1978, 14 (05) :367-373
[4]   METABOLISM OF MORPHINE AND HEROIN IN MAN [J].
BOERNER, U ;
ABBOTT, S ;
ROE, RL .
DRUG METABOLISM REVIEWS, 1975, 4 (01) :39-73
[5]   COMPARISON OF THE INVIVO AND INVITRO RATES OF FORMATION OF THE 3 MAIN OXIDATIVE METABOLITES OF ANTIPYRINE IN MAN [J].
BOOBIS, AR ;
BRODIE, MJ ;
KAHN, GC ;
TOVERUD, EL ;
BLAIR, IA ;
MURRAY, S ;
DAVIES, DS .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 12 (06) :771-777
[6]  
BRUNK SF, 1974, CLIN PHARMACOL THER, V16, P51
[7]   PHARMACOKINETIC INTERPRETATION OF THE ENTEROHEPATIC RECIRCULATION AND 1ST-PASS ELIMINATION OF MORPHINE IN THE RAT [J].
DAHLSTROM, BE ;
PAALZOW, LK .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1978, 6 (06) :505-519
[8]  
IWAMOTO K, 1977, J PHARMACOL EXP THER, V200, P236
[9]  
MAHON WA, 1977, CLIN PHARMACOL THER, V22, P228
[10]   MANAGEMENT OF INTRACTABLE PAIN IN PATIENTS WITH ADVANCED MALIGNANT DISEASE [J].
MOUNT, BM ;
MELZACK, R ;
MACKINNON, KJ .
JOURNAL OF UROLOGY, 1978, 120 (06) :720-725