ISOLATION OF HUMAN HEPATIC MICROSOMES AND THEIR INHIBITION BY CIMETIDINE AND RANITIDINE

被引:43
作者
HOENSCH, HP [1 ]
HUTZEL, H [1 ]
KIRCH, W [1 ]
OHNHAUS, EE [1 ]
机构
[1] UNIV ESSEN GESAMTHSCH, MED KLIN, HUFELANDSTR 55, D-4300 ESSEN 1, FED REP GER
关键词
D O I
10.1007/BF00547422
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:199 / 206
页数:8
相关论文
共 39 条
[1]  
AHMAD N, 1977, J PHARMACOL EXP THER, V203, P397
[2]  
BAHR VC, 1980, CLIN PHARMACOL THER, V27, P711
[3]  
Bell J A, 1981, Biochem Soc Trans, V9, P113
[4]  
BISSWANGER H, 1979, THEORIE METHODEN ENZ, P55
[5]   MONO-OXYGENASE ACTIVITY OF HUMAN-LIVER IN MICROSOMAL FRACTIONS OF NEEDLE-BIOPSY SPECIMENS [J].
BOOBIS, AR ;
BRODIE, MJ ;
KAHN, GC ;
FLETCHER, DR ;
SAUNDERS, JH ;
DAVIES, DS .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (01) :11-19
[6]   BIPHASIC O-DEETHYLATION OF PHENACETIN AND 7-ETHOXYCOUMARIN BY HUMAN AND RAT-LIVER MICROSOMAL FRACTIONS [J].
BOOBIS, AR ;
KAHN, GC ;
WHYTE, C ;
BRODIE, MJ ;
DAVIES, DS .
BIOCHEMICAL PHARMACOLOGY, 1981, 30 (17) :2451-2456
[7]   EFFECTS OF CIMETIDINE AND RANITIDINE ON HEPATIC DRUG-METABOLISM [J].
BREEN, KJ ;
BURY, R ;
DESMOND, PV ;
MASHFORD, ML ;
MORPHETT, B ;
WESTWOOD, B ;
SHAW, RG .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1982, 31 (03) :297-300
[8]   DRUG-METABOLISM IN LIVER-DISEASE - ACTIVITY OF HEPATIC MICROSOMAL METABOLIZING ENZYMES [J].
FARRELL, GC ;
COOKSLEY, WGE ;
POWELL, LW .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1979, 26 (04) :483-492
[9]   RANITIDINE BIOAVAILABILITY AND KINETICS IN NORMAL-MALE SUBJECTS [J].
GARG, DC ;
WEIDLER, DJ ;
ESHELMAN, FN .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1983, 33 (04) :445-452
[10]  
HAEGARTY AM, 1982, BMJ-BRIT MED J, V284, P1304