DIETHYL 3,6-DIHYDRO-2,4-DIMETHYL-2,6-METHANO-1,3-BENZOTHIAZOCINE-5,11-DICARBOXYLATES AS CALCIUM ENTRY ANTAGONISTS - NEW CONFORMATIONALLY RESTRAINED ANALOGS OF HANTZSCH 1,4-DIHYDROPYRIDINES RELATED TO NITRENDIPINE AS PROBES FOR RECEPTOR-SITE CONFORMATIONE

被引:45
作者
BALDWIN, JJ
CLAREMON, DA
LUMMA, PK
MCCLURE, DE
ROSENTHAL, SA
WINQUIST, RJ
FAISON, EP
KACZOROWSKI, GJ
TRUMBLE, MJ
SMITH, GM
机构
[1] MERCK SHARP & DOHME RES LABS,W POINT,PA 19486
[2] MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
关键词
D O I
10.1021/jm00387a019
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:690 / 695
页数:6
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