COCAETHYLENE INHIBITS DOPAMINE UPTAKE AND PRODUCES COCAINE-LIKE ACTIONS IN DRUG DISCRIMINATION STUDIES

被引:64
作者
WOODWARD, JJ [1 ]
MANSBACH, R [1 ]
CARROLL, FI [1 ]
BALSTER, RL [1 ]
机构
[1] RES TRIANGLE INST,RES TRIANGLE PK,NC 27709
关键词
D O I
10.1016/0014-2999(91)90531-T
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:235 / 236
页数:2
相关论文
共 5 条
[1]   COCAETHYLENE - A UNIQUE COCAINE METABOLITE DISPLAYS HIGH-AFFINITY FOR THE DOPAMINE TRANSPORTER [J].
HEARN, WL ;
FLYNN, DD ;
HIME, GW ;
ROSE, S ;
COFINO, JC ;
MANTEROATIENZA, E ;
WETLI, CV ;
MASH, DC .
JOURNAL OF NEUROCHEMISTRY, 1991, 56 (02) :698-701
[2]   COCAINE INHIBITION OF LIGAND-BINDING AT DOPAMINE, NOREPINEPHRINE AND SEROTONIN TRANSPORTERS - A STRUCTURE-ACTIVITY STUDY [J].
RITZ, MC ;
CONE, EJ ;
KUHAR, MJ .
LIFE SCIENCES, 1990, 46 (09) :635-645
[3]   PHENCYCLIDINE-LIKE DISCRIMINATIVE STIMULUS PROPERTIES OF MK-801 IN RATS [J].
WILLETTS, J ;
BALSTER, RL .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 146 (01) :167-169
[4]   CALCIUM-DEPENDENT AND CALCIUM-INDEPENDENT RELEASE OF ENDOGENOUS DOPAMINE FROM RAT STRIATAL SYNAPTOSOMES [J].
WOODWARD, JJ ;
CHANDLER, LJ ;
LESLIE, SW .
BRAIN RESEARCH, 1988, 473 (01) :91-98
[5]   DOPAMINE UPTAKE DURING FAST-PHASE ENDOGENOUS DOPAMINE RELEASE FROM MOUSE STRIATAL SYNAPTOSOMES [J].
WOODWARD, JJ ;
WILCOX, RE ;
LESLIE, SW ;
RIFFEE, WH .
NEUROSCIENCE LETTERS, 1986, 71 (01) :106-112