ADENOSINE 5'-(2-FLUORODIPHOSPHATE) IS A SELECTIVE AGONIST AT P2-PURINOCEPTORS MEDIATING RELAXATION OF SMOOTH-MUSCLE

被引:32
作者
HOURANI, SMO [1 ]
WELFORD, LA [1 ]
LOIZOU, GD [1 ]
CUSAK, NJ [1 ]
机构
[1] UNIV LONDON KINGS COLL,DEPT PHARMACOL,LONDON WC2R 2LS,ENGLAND
关键词
D O I
10.1016/0014-2999(88)90642-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:131 / 136
页数:6
相关论文
共 16 条
[1]  
Bumstock G, 1978, CELL MEMBRANE RECEPT, P107
[2]   IS THERE A BASIS FOR DISTINGUISHING 2 TYPES OF P2-PURINOCEPTOR [J].
BURNSTOCK, G ;
KENNEDY, C .
GENERAL PHARMACOLOGY, 1985, 16 (05) :433-440
[3]   STUDIES ON THE STEREOSELECTIVITY OF THE P2-PURINOCEPTOR [J].
BURNSTOCK, G ;
CUSACK, NJ ;
HILLS, JM ;
MACKENZIE, I ;
MEGHJI, P .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :907-913
[4]   SOME PHARMACOLOGICAL AND BIOCHEMICAL INTERACTIONS OF THE ENANTIOMERS OF ADENYLYL 5'-(BETA,GAMMA-METHYLENE)-DIPHOSPHONATE WITH THE GUINEA-PIG URINARY-BLADDER [J].
CUSACK, NJ ;
HOURANI, SMO .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 82 (01) :155-159
[5]   PHARMACOLOGICAL EFFECTS OF ISOPOLAR PHOSPHONATE ANALOGS OF ATP ON P-2-PURINOCEPTORS IN GUINEA-PIG TAENIA-COLI AND URINARY-BLADDER [J].
CUSACK, NJ ;
HOURANI, SMO ;
LOIZOU, GD ;
WELFORD, LA .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 90 (04) :791-795
[6]  
CUSACK NJ, 1979, BRIT J PHARMACOL, V67, P153
[7]   EXTRACELLULAR ATP - EFFECTS, SOURCES AND FATE [J].
GORDON, JL .
BIOCHEMICAL JOURNAL, 1986, 233 (02) :309-319
[8]   GAMMA-FLUOROADENOSINE TRIPHOSPHATE - SYNTHESIS, PROPERTIES, AND INTERACTION WITH MYOSIN AND HEAVY MEROMYOSIN [J].
HALEY, B ;
YOUNT, RG .
BIOCHEMISTRY, 1972, 11 (15) :2863-&
[9]   PHARMACOLOGICAL EFFECTS OF L-AMP-PCP ON ATP RECEPTORS IN SMOOTH-MUSCLE [J].
HOURANI, SMO ;
LOIZOU, GD ;
CUSACK, NJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 131 (01) :99-103
[10]   L-AMP-PCP, AN ATP RECEPTOR AGONIST IN GUINEA-PIG BLADDER, IS INACTIVE ON TAENIA-COLI [J].
HOURANI, SMO ;
WELFORD, LA ;
CUSACK, NJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 108 (02) :197-200