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SYNTHESIS OF DUAL ACTIVITY MOLECULES WITH THROMBOXANE ANTAGONIST AND THROMBOXANE SYNTHASE INHIBITORY ACTIVITY
被引:1
作者
:
RUSSELL, K
论文数:
0
引用数:
0
h-index:
0
机构:
ICI PHARMACEUT PLC,RES DEPT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI PHARMACEUT PLC,RES DEPT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
RUSSELL, K
[
1
]
GASKIN, H
论文数:
0
引用数:
0
h-index:
0
机构:
ICI PHARMACEUT PLC,RES DEPT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
ICI PHARMACEUT PLC,RES DEPT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
GASKIN, H
[
1
]
机构
:
[1]
ICI PHARMACEUT PLC,RES DEPT,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
来源
:
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
|
1992年
/ 2卷
/ 09期
关键词
:
D O I
:
10.1016/S0960-894X(00)80602-2
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
The synthesis of a series of dual acting thromboxane antagonist/thromboxane synthase inhibitors from a key tetrahydrocarbazole phenol is described.
引用
收藏
页码:985 / 986
页数:2
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YANG, ZY
[J].
TETRAHEDRON LETTERS,
1986,
27
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GUINDON Y, 1987, Patent No. 234708
[3]
N-(HETEROCYCLIC ALKYL)PYRIDO[2,1-B]QUINAZOLINE-8-CARBOXAMIDES AS ORALLY ACTIVE ANTIALLERGY AGENTS
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[J].
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: 185
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共 3 条
[1]
PALLADIUM-CATALYZED REACTION OF PHENYL FLUOROALKANESULFONATES WITH ALKYNES AND ALKENES
CHEN, QY
论文数:
0
引用数:
0
h-index:
0
CHEN, QY
YANG, ZY
论文数:
0
引用数:
0
h-index:
0
YANG, ZY
[J].
TETRAHEDRON LETTERS,
1986,
27
(10)
: 1171
-
1174
[2]
GUINDON Y, 1987, Patent No. 234708
[3]
N-(HETEROCYCLIC ALKYL)PYRIDO[2,1-B]QUINAZOLINE-8-CARBOXAMIDES AS ORALLY ACTIVE ANTIALLERGY AGENTS
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0
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TOBIAS, LD
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论文数:
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引用数:
0
h-index:
0
机构:
HOFFMANN LA ROCHE INC,DEPT PHARMACOL & CHEMOTHERAPY,NUTLEY,NJ 07110
HOFFMANN LA ROCHE INC,DEPT PHARMACOL & CHEMOTHERAPY,NUTLEY,NJ 07110
ODONNELL, M
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1987,
30
(01)
: 185
-
193
←
1
→