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ESTER BIO-ISOSTERES - SYNTHESIS OF OXADIAZOLYL-1-AZABICYCLO[2.2.1]HEPTANES AS MUSCARINIC AGONISTS
被引:56
作者
:
SAUNDERS, J
论文数:
0
引用数:
0
h-index:
0
SAUNDERS, J
MACLEOD, AM
论文数:
0
引用数:
0
h-index:
0
MACLEOD, AM
MERCHANT, K
论文数:
0
引用数:
0
h-index:
0
MERCHANT, K
SHOWELL, GA
论文数:
0
引用数:
0
h-index:
0
SHOWELL, GA
SNOW, RJ
论文数:
0
引用数:
0
h-index:
0
SNOW, RJ
STREET, LJ
论文数:
0
引用数:
0
h-index:
0
STREET, LJ
BAKER, R
论文数:
0
引用数:
0
h-index:
0
BAKER, R
机构
:
来源
:
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS
|
1988年
/ 24期
关键词
:
D O I
:
10.1039/c39880001618
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
引用
收藏
页码:1618 / 1619
页数:2
相关论文
共 10 条
[1]
PHYSOSTIGMINE AND ARECOLINE - EFFECTS OF INTRAVENOUS INFUSIONS IN ALZHEIMER PRESENILE-DEMENTIA
CHRISTIE, JE
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0
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CHRISTIE, JE
SHERING, A
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SHERING, A
FERGUSON, J
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0
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0
FERGUSON, J
GLEN, AIM
论文数:
0
引用数:
0
h-index:
0
GLEN, AIM
[J].
BRITISH JOURNAL OF PSYCHIATRY,
1981,
138
(JAN)
: 46
-
50
[2]
RELATIVE AFFINITIES OF DRUGS ACTING AT CHOLINOCEPTORS IN DISPLACING AGONIST AND ANTAGONIST RADIOLIGANDS - THE NMS OXO-M RATIO AS AN INDEX OF EFFICACY AT CORTICAL MUSCARINIC RECEPTORS
FREEDMAN, SB
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0
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FREEDMAN, SB
HARLEY, EA
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0
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0
HARLEY, EA
IVERSEN, LL
论文数:
0
引用数:
0
h-index:
0
IVERSEN, LL
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1988,
93
(02)
: 437
-
445
[3]
UNTERSUCHUNGEN IN DER CHINUCLIDIN-REIHE .3. 3-CHINUCLIDIN-CARBONSAURE
GROB, CA
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0
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0
h-index:
0
GROB, CA
RENK, E
论文数:
0
引用数:
0
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0
RENK, E
[J].
HELVETICA CHIMICA ACTA,
1954,
37
(06)
: 1689
-
1698
[4]
CHOLINERGIC APPROACHES TO THE TREATMENT OF ALZHEIMERS-DISEASE
HOLLANDER, E
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
HOLLANDER, E
MOHS, RC
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0
引用数:
0
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机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
MOHS, RC
DAVIS, KL
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0
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0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
DAVIS, KL
[J].
BRITISH MEDICAL BULLETIN,
1986,
42
(01)
: 97
-
100
[5]
KENAKIN TP, 1984, PHARMACOL REV, V36, P615
[6]
NIESCHUL.O, 1968, ARZNEI-FORSCHUNG, V18, P222
[7]
THE CHOLINERGIC HYPOTHESIS - 10 YEARS ON
PERRY, EK
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0
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PERRY, EK
[J].
BRITISH MEDICAL BULLETIN,
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[8]
2-METHYL-1,3-DIOXAAZASPIRO[4.5]DECANES AS NOVEL MUSCARINIC CHOLINERGIC AGONISTS
SAUNDERS, J
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MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
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SHOWELL, GA
SNOW, RJ
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MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
SNOW, RJ
BAKER, R
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MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
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HARLEY, EA
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MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
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FREEDMAN, SB
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MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
FREEDMAN, SB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1988,
31
(02)
: 486
-
491
[9]
RECOGNITION OF CHOLINERGIC AGONISTS BY THE MUSCARINIC RECEPTOR .1. ACETYLCHOLINE AND OTHER AGONISTS WITH THE NCCOCC BACKBONE
SCHULMAN, JM
论文数:
0
引用数:
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h-index:
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机构:
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
SCHULMAN, JM
SABIO, ML
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CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
SABIO, ML
DISCH, RL
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0
机构:
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
DISCH, RL
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
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(06)
: 817
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AZABICYCLIC ALCOHOLS .6. STEREOSPECIFIC SYNTHESIS OF 1-AZABICYLO[2.2.1]HEPTAN-3-OL EPIMERS
SPRY, DO
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SPRY, DO
AARON, HS
论文数:
0
引用数:
0
h-index:
0
机构:
Chemical Research Laboratory, Maryland 21010, Edgewood Arsenal
AARON, HS
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1969,
34
(11)
: 3674
-
&
←
1
→
共 10 条
[1]
PHYSOSTIGMINE AND ARECOLINE - EFFECTS OF INTRAVENOUS INFUSIONS IN ALZHEIMER PRESENILE-DEMENTIA
CHRISTIE, JE
论文数:
0
引用数:
0
h-index:
0
CHRISTIE, JE
SHERING, A
论文数:
0
引用数:
0
h-index:
0
SHERING, A
FERGUSON, J
论文数:
0
引用数:
0
h-index:
0
FERGUSON, J
GLEN, AIM
论文数:
0
引用数:
0
h-index:
0
GLEN, AIM
[J].
BRITISH JOURNAL OF PSYCHIATRY,
1981,
138
(JAN)
: 46
-
50
[2]
RELATIVE AFFINITIES OF DRUGS ACTING AT CHOLINOCEPTORS IN DISPLACING AGONIST AND ANTAGONIST RADIOLIGANDS - THE NMS OXO-M RATIO AS AN INDEX OF EFFICACY AT CORTICAL MUSCARINIC RECEPTORS
FREEDMAN, SB
论文数:
0
引用数:
0
h-index:
0
FREEDMAN, SB
HARLEY, EA
论文数:
0
引用数:
0
h-index:
0
HARLEY, EA
IVERSEN, LL
论文数:
0
引用数:
0
h-index:
0
IVERSEN, LL
[J].
BRITISH JOURNAL OF PHARMACOLOGY,
1988,
93
(02)
: 437
-
445
[3]
UNTERSUCHUNGEN IN DER CHINUCLIDIN-REIHE .3. 3-CHINUCLIDIN-CARBONSAURE
GROB, CA
论文数:
0
引用数:
0
h-index:
0
GROB, CA
RENK, E
论文数:
0
引用数:
0
h-index:
0
RENK, E
[J].
HELVETICA CHIMICA ACTA,
1954,
37
(06)
: 1689
-
1698
[4]
CHOLINERGIC APPROACHES TO THE TREATMENT OF ALZHEIMERS-DISEASE
HOLLANDER, E
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
HOLLANDER, E
MOHS, RC
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
MOHS, RC
DAVIS, KL
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PSYCHIAT,NEW YORK,NY 10029
DAVIS, KL
[J].
BRITISH MEDICAL BULLETIN,
1986,
42
(01)
: 97
-
100
[5]
KENAKIN TP, 1984, PHARMACOL REV, V36, P615
[6]
NIESCHUL.O, 1968, ARZNEI-FORSCHUNG, V18, P222
[7]
THE CHOLINERGIC HYPOTHESIS - 10 YEARS ON
PERRY, EK
论文数:
0
引用数:
0
h-index:
0
PERRY, EK
[J].
BRITISH MEDICAL BULLETIN,
1986,
42
(01)
: 63
-
69
[8]
2-METHYL-1,3-DIOXAAZASPIRO[4.5]DECANES AS NOVEL MUSCARINIC CHOLINERGIC AGONISTS
SAUNDERS, J
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
SAUNDERS, J
SHOWELL, GA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
SHOWELL, GA
SNOW, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
SNOW, RJ
BAKER, R
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
BAKER, R
HARLEY, EA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
HARLEY, EA
FREEDMAN, SB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
MERCK SHARP & DOHME RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
FREEDMAN, SB
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1988,
31
(02)
: 486
-
491
[9]
RECOGNITION OF CHOLINERGIC AGONISTS BY THE MUSCARINIC RECEPTOR .1. ACETYLCHOLINE AND OTHER AGONISTS WITH THE NCCOCC BACKBONE
SCHULMAN, JM
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
SCHULMAN, JM
SABIO, ML
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
SABIO, ML
DISCH, RL
论文数:
0
引用数:
0
h-index:
0
机构:
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
CUNY MT SINAI SCH MED,DEPT PHARMACOL,NEW YORK,NY 10029
DISCH, RL
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1983,
26
(06)
: 817
-
823
[10]
AZABICYCLIC ALCOHOLS .6. STEREOSPECIFIC SYNTHESIS OF 1-AZABICYLO[2.2.1]HEPTAN-3-OL EPIMERS
SPRY, DO
论文数:
0
引用数:
0
h-index:
0
机构:
Chemical Research Laboratory, Maryland 21010, Edgewood Arsenal
SPRY, DO
AARON, HS
论文数:
0
引用数:
0
h-index:
0
机构:
Chemical Research Laboratory, Maryland 21010, Edgewood Arsenal
AARON, HS
[J].
JOURNAL OF ORGANIC CHEMISTRY,
1969,
34
(11)
: 3674
-
&
←
1
→