OCTAPEPTIDE ANALOGS OF SOMATOSTATIN EXHIBITING GREATLY ENHANCED INVIVO AND INVITRO INHIBITION OF GROWTH-HORMONE SECRETION IN THE RAT

被引:54
作者
MURPHY, WA
HEIMAN, ML
LANCE, VA
MEZO, I
COY, DH
机构
关键词
D O I
10.1016/0006-291X(85)91895-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:922 / 928
页数:7
相关论文
共 19 条
[1]  
BAUER W, 1982, LIFE SCI, V31, P1133, DOI 10.1016/0024-3205(82)90087-X
[2]  
COY DH, 1985, SOMATOSTATIN, P325
[3]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[4]  
FREIDINGER RM, 1983, PEPTIDES STRUCTURE F, P349
[5]   AN EXTREMELY SENSITIVE INVITRO MODEL FOR ELUCIDATING STRUCTURE-ACTIVITY-RELATIONSHIPS OF GROWTH HORMONE-RELEASING FACTOR ANALOGS [J].
HEIMAN, ML ;
NEKOLA, MV ;
MURPHY, WA ;
LANCE, VA ;
COY, DH .
ENDOCRINOLOGY, 1985, 116 (01) :410-415
[6]   ADMINISTRATION OF HUMAN PANCREATIC GROWTH HORMONE-RELEASING FACTOR (GRF) ANALOGS ENHANCES RESPONSIVENESS OF CULTURED RAT PITUITARY-CELLS TO GRF [J].
HEIMAN, ML ;
MURPHY, WA ;
NEKOLA, MV ;
LANCE, VA ;
COY, DH .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 124 (01) :217-222
[7]   EFFECT OF LONG-ACTING SOMATOSTATIN-ANALOGUE, SMS 201995, ON GUT HORMONE-SECRETION IN NORMAL SUBJECTS [J].
KRAENZLIN, ME ;
WOOD, SM ;
NEUFELD, M ;
ADRIAN, TE ;
BLOOM, SR .
EXPERIENTIA, 1985, 41 (06) :738-740
[8]   OPIATE ANTAGONISTIC PROPERTIES OF AN OCTAPEPTIDE SOMATOSTATIN ANALOG [J].
MAURER, R ;
GAEHWILER, BH ;
BUESCHER, HH ;
HILL, RC ;
ROEMER, D .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (15) :4815-4817
[9]   POTENT, HIGHLY SELECTIVE-INHIBITION OF GROWTH-HORMONE SECRETION BY POSITION 4 SOMATOSTATIN ANALOGS [J].
MURPHY, WA ;
MEYERS, CA ;
COY, DH .
ENDOCRINOLOGY, 1981, 109 (02) :491-495
[10]   CONFORMATIONALLY RESTRICTED ANALOGS OF SOMATOSTATIN WITH HIGH MU-OPIATE RECEPTOR SPECIFICITY [J].
PELTON, JT ;
GULYA, K ;
HRUBY, VJ ;
DUCKLES, SP ;
YAMAMURA, HI .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (01) :236-239