DESIGN AND SYNTHESIS OF SOMATOSTATIN ANALOGS WITH TOPOGRAPHICAL PROPERTIES THAT LEAD TO HIGHLY POTENT AND SPECIFIC MU-OPIOID RECEPTOR ANTAGONISTS WITH GREATLY REDUCED BINDING AT SOMATOSTATIN RECEPTORS

被引：126

作者：

KAZMIERSKI, W

WIRE, WS

LUI, GK

KNAPP, RJ

SHOOK, JE

BURKS, TF

YAMAMURA, HI

HRUBY, VJ

机构：

[1] UNIV ARIZONA,DEPT CHEM,TUCSON,AZ 85721

[2] UNIV ARIZONA,DEPT PHARMACOL,TUCSON,AZ 85721

来源：

关键词：

D O I：

10.1021/jm00119a019

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2170 / 2177

页数：8

共 35 条

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