PEPTIDE-E - OPIATE RECEPTOR-BINDING PROFILE IN THE RAT-BRAIN MEMBRANE ASSAY - COMPARISON WITH BETA-ENDORPHIN

被引:4
作者
WESTPHAL, M [1 ]
LI, CH [1 ]
HEIMER, EP [1 ]
MEIENHOFER, J [1 ]
机构
[1] HOFFMANN LA ROCHE INC,ROCHE RES CTR,DEPT BIOORGAN CHEM,NUTLEY,NJ 07110
关键词
D O I
10.1016/0006-291X(83)90673-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1084 / 1088
页数:5
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共 14 条
[1]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[2]  
FERRARA P, 1980, INT J PEPT PROT RES, V16, P66
[3]   SPECTRUM OF THE MU-BINDING, DELTA-BINDING AND KAPPA-BINDING SITES IN HOMOGENATES OF RAT-BRAIN [J].
GILLAN, MGC ;
KOSTERLITZ, HW .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (03) :461-468
[4]  
HAMMONDS RG, 1982, INT J PEPT PROT RES, V19, P556
[5]  
HEIMER EP, 1983, ARCH BIOCH BIOPHYS, V225
[6]   MULTIPLE ENDOGENOUS OPIOID-PEPTIDES [J].
HOLLT, V .
TRENDS IN NEUROSCIENCES, 1983, 6 (01) :24-26
[7]   OPIOID-PEPTIDES DERIVED FROM PRO-ENKEPHALIN A BUT NOT THAT FROM PRO-ENKEPHALIN-B ARE SUBSTANTIAL ANALGESICS AFTER ADMINISTRATION INTO BRAIN OF MICE [J].
HOLLT, V ;
TULUNAY, FC ;
WOO, SK ;
LOH, HH ;
HERZ, A .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 85 (3-4) :355-356
[8]  
HOUGHTEN RA, 1980, INT J PEPT PROT RES, V16, P311
[9]   A HIGHLY POTENT 3200-DALTON ADRENAL OPIOID PEPTIDE THAT CONTAINS BOTH A [MET]-ENKEPHALIN AND [LEU]ENKEPHALIN SEQUENCE [J].
KILPATRICK, DL ;
TANIGUCHI, T ;
JONES, BN ;
STERN, AS ;
SHIVELY, JE ;
HULLIHAN, J ;
KIMURA, S ;
STEIN, S ;
UDENFRIEND, S .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (05) :3265-3268
[10]   SYNTHESIS AND ANALGESIC ACTIVITY OF HUMAN BETA-ENDORPHIN [J].
LI, CH ;
YAMASHIRO, D ;
TSENG, LF ;
LOH, HH .
JOURNAL OF MEDICINAL CHEMISTRY, 1977, 20 (03) :325-328