SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 3-AMINOMETHYL-1,2-DITHILANE AND 4-AMINOMETHYL-1,2-DITHIOLANE

被引：8

作者：

UNEME, H

MITSUDERA, H

YAMADA, J

KAMIKADO, T

KONO, Y

MANABE, Y

NUMATA, M

机构：

[1] Agricultural Research Laboratories, Agro Division, Takeda Chemical Industries Ltd., Ibaraki 300-42, 10 Wadai, Tsukuba

[2] Department of Medical Entomology, National Institute of Health, Tokyo 141, 2-10-35 Kamiosaki, Shinagawa-ku

来源：

BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY | 1992年 / 56卷 / 08期

关键词：

BRP; brown rice planthoppers; CCW; common cutworms; NHM; northern house mosquito larvae; NTX; nereistoxin; RSB; rice stem borers; TSM; two-spotted spider mites;

D O I：

10.1271/bbb.56.1293

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

The structures of the insecticidal alkaloids, guinesines (4-hydroxy-3-(1-methyl-2-pyrrolidinyl)-1,2-dithiolanes), were simplified in several ways while retaining the dithiolane ring. Most of the compounds synthesized showed activity against Chilo suppressalis and Tetranychus urticae. High potency against Chilo suppressalis was displayed by 3-(dimethylaminomethyl)-1,2-dithiolane, and a broad pesticidal spectrum was recognized in the case of 4-(dimethylaminomethyl)-1,2-dithiolane.

引用

页码：1293 / 1299

页数：7

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