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ACTINOPLANIC-ACID-A - A MACROCYCLIC POLYCARBOXYLIC ACID WHICH IS A POTENT INHIBITOR OF RAS FARNESYL-PROTEIN TRANSFERASE
被引:28
作者
:
SINGH, SB
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
SINGH, SB
LIESCH, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
LIESCH, JM
LINGHAM, RB
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
LINGHAM, RB
GOETZ, MA
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
GOETZ, MA
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
机构:
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
GIBBS, JB
机构
:
[1]
Merck Research Laboratories, Rahway, New Jersey, P.O. Box 2000
[2]
West Point
来源
:
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
|
1994年
/ 116卷
/ 25期
关键词
:
D O I
:
10.1021/ja00104a066
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
[No abstract available]
引用
收藏
页码:11606 / 11607
页数:2
相关论文
共 19 条
[1]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[2]
STRUCTURE ELUCIDATION OF THE FUMONISINS, MYCOTOXINS FROM FUSARIUM-MONILIFORME
BEZUIDENHOUT, SC
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
BEZUIDENHOUT, SC
GELDERBLOM, WCA
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
GELDERBLOM, WCA
GORSTALLMAN, CP
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
GORSTALLMAN, CP
HORAK, RM
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
HORAK, RM
MARASAS, WFO
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
MARASAS, WFO
SPITELLER, G
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
SPITELLER, G
VLEGGAAR, R
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
VLEGGAAR, R
[J].
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS,
1988,
(11)
: 743
-
745
[3]
P21RAS IS MODIFIED BY A FARNESYL ISOPRENOID
CASEY, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
CASEY, PJ
SOLSKI, PA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
SOLSKI, PA
DER, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
DER, CJ
BUSS, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
BUSS, JE
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(21)
: 8323
-
8327
[4]
DER CJ, 1991, CANCER CELL-MON REV, V3, P331
[5]
Gibbs J B, 1992, Semin Cancer Biol, V3, P383
[6]
RAS C-TERMINAL PROCESSING ENZYMES - MINIREVIEW NEW DRUG TARGETS
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
[J].
CELL,
1991,
65
(01)
: 1
-
4
[7]
GIBBS JB, 1993, J BIOL CHEM, V268, P7617
[8]
FARNESYLTRANSFERASE INHIBITORS - RAS RESEARCH YIELDS A POTENTIAL CANCER THERAPEUTIC
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
OLIFF, A
论文数:
0
引用数:
0
h-index:
0
OLIFF, A
KOHL, NE
论文数:
0
引用数:
0
h-index:
0
KOHL, NE
[J].
CELL,
1994,
77
(02)
: 175
-
178
[9]
JAMES GJ, 1993, SCIENCE, V260, P197
[10]
SELECTIVE-INHIBITION OF RAS-DEPENDENT TRANSFORMATION BY A FARNESYLTRANSFERASE INHIBITOR
KOHL, NE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
KOHL, NE
MOSSER, SD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
MOSSER, SD
DESOLMS, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
DESOLMS, SJ
GIULIANI, EA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GIULIANI, EA
POMPLIANO, DL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
POMPLIANO, DL
GRAHAM, SL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GRAHAM, SL
SMITH, RL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
SMITH, RL
SCOLNICK, EM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
SCOLNICK, EM
OLIFF, A
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
OLIFF, A
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GIBBS, JB
[J].
SCIENCE,
1993,
260
(5116)
: 1934
-
1937
←
1
2
→
共 19 条
[1]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[2]
STRUCTURE ELUCIDATION OF THE FUMONISINS, MYCOTOXINS FROM FUSARIUM-MONILIFORME
BEZUIDENHOUT, SC
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
BEZUIDENHOUT, SC
GELDERBLOM, WCA
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
GELDERBLOM, WCA
GORSTALLMAN, CP
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
GORSTALLMAN, CP
HORAK, RM
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
HORAK, RM
MARASAS, WFO
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
MARASAS, WFO
SPITELLER, G
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
SPITELLER, G
VLEGGAAR, R
论文数:
0
引用数:
0
h-index:
0
机构:
CSIR, NATL CHEM RES LAB, POB 395, PRETORIA 0001, SOUTH AFRICA
VLEGGAAR, R
[J].
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS,
1988,
(11)
: 743
-
745
[3]
P21RAS IS MODIFIED BY A FARNESYL ISOPRENOID
CASEY, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
CASEY, PJ
SOLSKI, PA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
SOLSKI, PA
DER, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
DER, CJ
BUSS, JE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV TEXAS,SW MED CTR,DEPT PHARMACOL,5323 HARRY HINES BLVD,DALLAS,TX 75235
BUSS, JE
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(21)
: 8323
-
8327
[4]
DER CJ, 1991, CANCER CELL-MON REV, V3, P331
[5]
Gibbs J B, 1992, Semin Cancer Biol, V3, P383
[6]
RAS C-TERMINAL PROCESSING ENZYMES - MINIREVIEW NEW DRUG TARGETS
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
[J].
CELL,
1991,
65
(01)
: 1
-
4
[7]
GIBBS JB, 1993, J BIOL CHEM, V268, P7617
[8]
FARNESYLTRANSFERASE INHIBITORS - RAS RESEARCH YIELDS A POTENTIAL CANCER THERAPEUTIC
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
OLIFF, A
论文数:
0
引用数:
0
h-index:
0
OLIFF, A
KOHL, NE
论文数:
0
引用数:
0
h-index:
0
KOHL, NE
[J].
CELL,
1994,
77
(02)
: 175
-
178
[9]
JAMES GJ, 1993, SCIENCE, V260, P197
[10]
SELECTIVE-INHIBITION OF RAS-DEPENDENT TRANSFORMATION BY A FARNESYLTRANSFERASE INHIBITOR
KOHL, NE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
KOHL, NE
MOSSER, SD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
MOSSER, SD
DESOLMS, SJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
DESOLMS, SJ
GIULIANI, EA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GIULIANI, EA
POMPLIANO, DL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
POMPLIANO, DL
GRAHAM, SL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GRAHAM, SL
SMITH, RL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
SMITH, RL
SCOLNICK, EM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
SCOLNICK, EM
OLIFF, A
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
OLIFF, A
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT CANC RES,W POINT,PA 19486
GIBBS, JB
[J].
SCIENCE,
1993,
260
(5116)
: 1934
-
1937
←
1
2
→