TRIMETREXATE - A 2ND GENERATION FOLATE ANTAGONIST IN CLINICAL-TRIAL

被引:58
作者
LIN, JT
BERTINO, JR
机构
[1] YALE UNIV,SCH MED,DEPT MED,NEW HAVEN,CT 06510
[2] YALE UNIV,SCH MED,DEPT PHARMACOL,NEW HAVEN,CT 06510
关键词
D O I
10.1200/JCO.1987.5.12.2032
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:2032 / 2040
页数:9
相关论文
共 68 条
  • [1] A RAPID AND SENSITIVE METHOD FOR DETERMINATION OF TRIMETREXATE FROM BIOLOGICAL-FLUIDS
    ACKERLY, CC
    HARTSHORN, J
    TONG, WP
    MCCORMACK, JJ
    [J]. JOURNAL OF LIQUID CHROMATOGRAPHY, 1985, 8 (01): : 125 - 134
  • [2] ALLEGRA CJ, 1986, 26TH INT C ANT ANT C, P224
  • [3] ANDERSON JA, 1983, RR74500565 WARN PARK
  • [4] ANDREWS L, 1985, P AM ASSOC CANC RES, V26, P370
  • [5] ARKIN H, 1986, P AM ASSOC CANC RES, V27, P269
  • [6] Baker BR, 1967, DESIGN ACTIVE SITE D
  • [7] BALIS FM, 1986, CANCER RES, V46, P169
  • [8] BALIS FM, 1987, P AM SOC CLIN ONCOL, V6, P154
  • [9] 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL]QUINAZOLINE (TMQ), A POTENT NON-CLASSICAL FOLATE ANTAGONIST INHIBITOR .1. EFFECT ON DIHYDROFOLATE-REDUCTASE AND GROWTH OF RODENT TUMORS INVITRO AND INVIVO
    BERTINO, JR
    SAWICKI, WL
    MOROSON, BA
    CASHMORE, AR
    ELSLAGER, EF
    [J]. BIOCHEMICAL PHARMACOLOGY, 1979, 28 (12) : 1983 - 1987
  • [10] BERTINO JR, 1977, P AM ASSOC CANC RES, V18, P168