CHARACTERIZATION OF FLUNITRAZEPAM AND BETA-CARBOLINE HIGH-AFFINITY BINDING IN BOVINE PINEAL-GLAND

被引:22
作者
LOWENSTEIN, PR [1 ]
CARDINALI, DP [1 ]
机构
[1] CTR ESTUDIOS FARMACOL & PRINCIPIOS NAT,SERRANO 665-669,RA-1414 BUENOS AIRES,ARGENTINA
关键词
D O I
10.1159/000123533
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:150 / 154
页数:5
相关论文
共 34 条
[1]   PROSTAGLANDINS-A AS POSSIBLE ENDOGENOUS LIGANDS OF BENZODIAZEPINE RECEPTOR [J].
ASANO, T ;
OGASAWARA, N .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 80 (2-3) :271-274
[2]   IDENTIFICATION OF INOSINE AND HYPOXANTHINE AS ENDOGENOUS LIGANDS FOR THE BRAIN BENZODIAZEPINE-BINDING SITES [J].
ASANO, T ;
SPECTOR, S .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (02) :977-981
[3]  
BENNETT JP, 1978, NEUROTRANSMITTER REC, P57
[4]   [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].
BRAESTRUP, C ;
NIELSEN, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) :333-341
[5]   URINARY AND BRAIN BETA-CARBOLINE-3-CARBOXYLATES AS POTENT INHIBITORS OF BRAIN BENZODIAZEPINE RECEPTORS [J].
BRAESTRUP, C ;
NIELSEN, M ;
OLSEN, CE .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (04) :2288-2292
[6]  
CHABOT G, 1982, J PHYSL PHARM, V60, P589
[7]   THE KINETICS OF NOREPINEPHRINE-INDUCED STIMULATION OF SEROTONIN N-ACETYLTRANSFERASE IN BOVINE PINEAL-GLAND [J].
CHAN, A ;
EBADI, M .
NEUROENDOCRINOLOGY, 1980, 31 (04) :244-251
[8]   IS THE BENZODIAZEPINE RECEPTOR COUPLED TO A CHLORIDE ANION CHANNEL [J].
COSTA, T ;
RODBARD, D ;
PERT, CB .
NATURE, 1979, 277 (5694) :315-317
[9]   ETHYL BETA-CARBOLINE CARBOXYLATE LOWERS SEIZURE THRESHOLD AND ANTAGONIZES FLURAZEPAM-INDUCED SEDATION IN RATS [J].
COWEN, PJ ;
GREEN, AR ;
NUTT, DJ ;
MARTIN, IL .
NATURE, 1981, 290 (5801) :54-55
[10]   CHARACTERISTICS OF GABA BINDING-SITES IN BOVINE PINEAL-GLAND [J].
EBADI, M ;
CHAN, A .
BRAIN RESEARCH BULLETIN, 1980, 5 :179-187