AN IMPROVED ENTRY TO A KEY INTERMEDIATE FOR THIENAMYCIN SYNTHESIS FROM METHYL (R)-3-HYDROXYBUTANOATE VIA DIRECT EPIMERIZATION AT C-3 ON 2-AZETIDINONE RINGS

被引：56

作者：

CHIBA, T ^{[1
]}

NAKAI, T ^{[1
]}

机构：

[1] TOKYO INST TECHNOL,DEPT CHEM TECHNOL,MEGURO KU,TOKYO 152,JAPAN

来源：

TETRAHEDRON LETTERS | 1985年 / 26卷 / 38期

关键词：

D O I：

10.1016/S0040-4039(00)98775-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：4647 / 4648

页数：2

共 9 条

[1] STEREOCONTROLLED TOTAL SYNTHESIS OF THE CHIRAL BUILDING BLOCK (3S,4R)-3-[(R)-1-HYDROXYETHYL]-4-ACETYLOXY-AZETIDIN-2-ONE - A USEFUL SYNTHON FOR THE SYNTHESIS OF (+)-THIENAMYCIN, CARBAPENEMS AND PENEMS
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[2] A SYNTHETIC APPROACH TO (+)-THIENAMYCIN FROM METHYL (R)-3-HYDROXYBUTANOATE - A NEW ENTRY TO (3R,4R)-3-[(R)-1-HYDROXYETHYL]-4-ACETOXY-2-AZETIDINONE
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[J]. CHEMISTRY LETTERS, 1985, (05) : 651 - 654
[3] A FACILE ENTRY TO 3-(1-HYDROXYETHYL)-2-AZETIDINONES FROM METHYL(R)-3-HYDROXYBUTANOATE BASED ON THE ESTER ENOLATE-ALDIMINE CONDENSATION
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[J]. CHEMISTRY LETTERS, 1984, (11) : 1927 - 1930
[4] CHIBA T, 1985, UNPUB 50TH ANN M CHE
[5] N-TRIMETHYLSILYL IMINES - APPLICATIONS TO THE SYNTHESIS OF BETA-LACTAMS
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[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1984, 106 (17) : 4819 - 4825
[6] STEREOCONTROLLED SYNTHESIS OF (+)-THIENAMYCIN FROM 3(R)-HYDROXYBUTYRIC ACID
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[J]. TETRAHEDRON LETTERS, 1985, 26 (12) : 1523 - 1526
[7] SYNTHESIS OF CARBAPENEM ANTIBIOTICS
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[J]. HETEROCYCLES, 1982, 17 : 463 - 506
[8] AN EFFICIENT SYNTHESIS OF 2-SUBSTITUTED-THIO-6-HYDROXYETHYL-PENEM-3-CARBOXYLIC ACIDS VIA 2-THIOXOPENAMS
LEANZA, WJ
DININNO, F
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CHRISTENSEN, BG
[J]. TETRAHEDRON, 1983, 39 (15) : 2505 - 2513
[9] SYNTHESIS OF 1-CARBAPENEMS AND 1-CARBAPENAMS
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[J]. JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN, 1983, 41 (01) : 62 - 76

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