ENOL LACTONE INHIBITORS OF SERINE PROTEASES - THE EFFECT OF REGIOCHEMISTRY ON THE INACTIVATION BEHAVIOR OF PHENYL-SUBSTITUTED (HALOMETHYLENE)TETRAHYDROPYRANONES AND -DIHYDROFURANONES AND (HALOMETHYLENE)TETRAHYDROPYRANONES TOWARD ALPHA-CHYMOTRYPSIN - STABLE ACYL ENZYME INTERMEDIATE

被引：38

作者：

SOFIA, MJ ^{[1
]}

KATZENELLENBOGEN, JA ^{[1
]}

机构：

[1] UNIV ILLINOIS,SCH CHEM SCI,URBANA,IL 61801

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 02期

关键词：

D O I：

10.1021/jm00152a011

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：230 / 238

页数：9

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