A -CH2CH-C+NR(2) SYNTHON - NOVEL PREPARATIONS OF 1,3-DISUBSTITUTED ALLYLAMINES AND OF 1,2-DIARYL PYRROLES

被引：24

作者：

KATRITZKY, AR

CHANG, HX

VERIN, SV

机构：

[1] Center for Heterocyclic Compounds, Department of Chemistry, University of Florida, Gainesville

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 03期

关键词：

D O I：

10.1016/0040-4039(94)02265-D

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1-(3-Morpholinoprop-2-enyl)benzotriazole (1) is a useful synthon of the type [(CH2)-C---CH=C(+)NR(2)] as demonstrated by the preparation of allylamines 4. It can also provide a [(+ -) CH-CH=CH+] fragment for the synthesis of 1,2-diarylpyrroles 6.

引用

页码：343 / 346

页数：4

共 15 条

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