STEREOSELECTIVE BLOCKADE AT [H-3]5-HT BINDING-SITES AND AT THE 5-HT AUTORECEPTOR BY PROPRANOLOL

被引:211
作者
MIDDLEMISS, DN
机构
关键词
D O I
10.1016/0014-2999(84)90173-0
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:289 / 293
页数:5
相关论文
共 10 条
[1]   EVIDENCE FOR COMMON PHARMACOLOGICAL PROPERTIES OF [H-3]5-HYDROXYTRYPTAMINE BINDING-SITES, PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE AUTORECEPTORS IN CNS AND INHIBITORY PRE-SYNAPTIC 5-HYDROXYTRYPTAMINE RECEPTORS ON SYMPATHETIC-NERVES [J].
ENGEL, G ;
GOTHERT, M ;
MULLERSCHWEINITZER, E ;
SCHLICKER, E ;
SISTONEN, L ;
STADLER, PA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 324 (02) :116-124
[2]   A CUMULATIVE DOSE-RESPONSE TECHNIQUE FOR THE CHARACTERIZATION OF PRE-SYNAPTIC RECEPTORS MODULATING [3H]NORADRENALIN RELEASE FROM RAT-BRAIN SLICES [J].
FRANKHUYZEN, AL ;
MULDER, AH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 78 (01) :91-97
[3]   AUTORECEPTOR-MEDIATED INHIBITION OF H-3-5-HYDROXYTRYPTAMINE RELEASE FROM RAT-BRAIN CORTEX SLICES BY ANALOGS OF 5-HYDROXYTRYPTAMINE [J].
GOTHERT, M ;
SCHLICKER, E .
LIFE SCIENCES, 1983, 32 (11) :1183-1191
[5]   COMPARISON OF THE PHARMACOLOGICAL CHARACTERISTICS OF 5-HT1 AND 5-HT2 BINDING-SITES WITH THOSE OF SEROTONIN AUTORECEPTORS WHICH MODULATE SEROTONIN RELEASE [J].
MARTIN, LL ;
SANDERSBUSH, E .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (03) :165-170
[6]   DIRECT EVIDENCE FOR AN INTERACTION OF BETA-ADRENERGIC BLOCKERS WITH 5-HT RECEPTOR [J].
MIDDLEMISS, DN ;
BLAKEBOROUGH, L ;
LEATHER, SR .
NATURE, 1977, 267 (5608) :289-290
[7]   8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)-TETRALIN DISCRIMINATES BETWEEN SUBTYPES OF THE 5-HT1 RECOGNITION SITE [J].
MIDDLEMISS, DN ;
FOZARD, JR .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 90 (01) :151-153
[8]  
MIDDLEMISS DN, 1983, NAUNYNSCHMIEDEB AR S, V324, P76
[9]  
NAHORSKI SR, 1983, BRIT J PHARMACOL, V78, P1071
[10]   DISCRIMINATION OF MULTIPLE [H-3]5-HYDROXYTRYPTAMINE BINDING-SITES BY THE NEUROLEPTIC SPIPERONE IN RAT-BRAIN [J].
PEDIGO, NW ;
YAMAMURA, HI ;
NELSON, DL .
JOURNAL OF NEUROCHEMISTRY, 1981, 36 (01) :220-226