MEPROADIFEN ENHANCES ACTIVATION AND DESENSITIZATION OF THE ACETYLCHOLINE RECEPTOR-IONIC CHANNEL COMPLEX (ACHR) - SINGLE CHANNEL STUDIES

被引:21
作者
ARACAVA, Y
ALBUQUERQUE, EX
机构
关键词
D O I
10.1016/0014-5793(84)81171-0
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
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页码:267 / 274
页数:8
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  • [1] AKAIKE A, 1984, MOL PHARMACOL, V25, P102
  • [2] ARACAVA Y, 1983, NEUR ABSTR, V9, P733
  • [3] ARACAVA Y, MOL PHARM
  • [4] ELECTRO-PHYSIOLOGICAL AND BIOCHEMICAL-STUDIES ON ENHANCEMENT OF DESENSITIZATION BY PHENOTHIAZINE NEUROLEPTICS
    CARP, JS
    ARONSTAM, RS
    WITKOP, B
    ALBUQUERQUE, EX
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (01): : 310 - 314
  • [5] IMPROVED PATCH-CLAMP TECHNIQUES FOR HIGH-RESOLUTION CURRENT RECORDING FROM CELLS AND CELL-FREE MEMBRANE PATCHES
    HAMILL, OP
    MARTY, A
    NEHER, E
    SAKMANN, B
    SIGWORTH, FJ
    [J]. PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1981, 391 (02): : 85 - 100
  • [6] MULTIPLE SITES OF ACTION FOR NONCOMPETITIVE BLOCKERS ON ACETYLCHOLINE-RECEPTOR RICH MEMBRANE-FRAGMENTS FROM TORPEDO-MARMORATA
    HEIDMANN, T
    OSWALD, RE
    CHANGEUX, JP
    [J]. BIOCHEMISTRY, 1983, 22 (13) : 3112 - 3127
  • [7] FAST KINETIC STUDIES ON THE ALLOSTERIC INTERACTIONS BETWEEN ACETYLCHOLINE-RECEPTOR AND LOCAL-ANESTHETIC BINDING-SITES
    HEIDMANN, T
    CHANGEUX, JP
    [J]. EUROPEAN JOURNAL OF BIOCHEMISTRY, 1979, 94 (01): : 281 - 296
  • [8] STABILIZATION OF THE HIGH-AFFINITY STATE OF THE MEMBRANE-BOUND ACETYLCHOLINE-RECEPTOR FROM TORPEDO-MARMORATA BY NONCOMPETITIVE BLOCKERS - EVIDENCE FOR DUAL INTERACTION AND PHARMACOLOGICAL SELECTIVITY
    HEIDMANN, T
    CHANGEUX, JP
    [J]. FEBS LETTERS, 1981, 131 (02): : 239 - 244
  • [9] ASYMMETRY OF THE ACETYLCHOLINE CHANNEL REVEALED BY QUATERNARY ANESTHETICS
    HORN, R
    BRODWICK, MS
    DICKEY, WD
    [J]. SCIENCE, 1980, 210 (4466) : 205 - 207
  • [10] IKEDA SR, MOL PHARM