AMINO PROTECTION USING TRIAZONES

被引：40

作者：

KNAPP, S

HALE, JJ

BASTOS, M

GIBSON, FS

机构：

[1] Department of Chemistry, Rutgers The State University of New Jersey, New Brunswick

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 15期

关键词：

D O I：

10.1016/0040-4039(90)80084-Y

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Primary amines protected by incorporation into a "triazone" derivative (3) are stable to various reduction, oxidation, organometallic, and basic hydrolysis conditions, and may be regenerated by treatment with aqueous ammonium chloride at 70 °. An application to polyamine synthesis is described. © 1990.

引用

页码：2109 / 2112

页数：4

共 30 条

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