GEM-DISUBSTITUTED AMINO-ETHER BASED SUBSTANCE-P ANTAGONISTS

被引:30
作者
HARRISON, T
WILLIAMS, BJ
SWAIN, CJ
机构
[1] Department of Medicinal Chemistry, Neuroscience Research Centre, Merck Sharp and Dohme Research Laboratories, Harlow, Essex CM20 2QR, Terlings Park, Eastwick Road
关键词
D O I
10.1016/S0960-894X(01)80585-0
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
The design and syntheses of new series of gem- disubstituted pyrrolidine and piperidine derivatives (eg. 2 and 3) is described.
引用
收藏
页码:2733 / 2734
页数:2
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[3]  
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YASUO H, 1979, CHEM PHARM BULL, V28, P1931