SYNTHESIS AND CHARACTERIZATION OF AN AFFINITY LABEL FOR BRAIN RECEPTORS TO PSYCHOTOMIMETIC BENZOMORPHANS - DIFFERENTIATION OF SIGMA-TYPE AND PHENCYCLIDINE RECEPTORS

被引:19
作者
ADAMS, JT
TEAL, PM
SONDERS, MS
TESTER, B
ESHERICK, JS
SCHERZ, MW
KEANA, JFW
WEBER, E
机构
[1] OREGON HLTH SCI UNIV,VOLLUM INST ADV BIOMED RES,PORTLAND,OR 97201
[2] OREGON HLTH SCI UNIV,DEPT BIOCHEM,PORTLAND,OR 97201
[3] OREGON HLTH SCI UNIV,DEPT PSYCHIAT,PORTLAND,OR 97201
[4] UNIV OREGON,DEPT CHEM,EUGENE,OR 97403
关键词
D O I
10.1016/0014-2999(87)90654-6
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:61 / 71
页数:11
相关论文
共 23 条
  • [1] PHENCYCLIDINE (PCP) - A REVIEW AND PERSPECTIVES
    ANILINE, O
    PITTS, FN
    [J]. CRC CRITICAL REVIEWS IN TOXICOLOGY, 1982, 10 (02): : 145 - 177
  • [2] BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
  • [3] GOLDSTEIN A, 1984, MOL PHARMACOL, V25, P343
  • [4] HAERTZEN C A, 1970, Psychopharmacologia, V18, P366, DOI 10.1007/BF00402763
  • [5] JAMES IF, 1984, MOL PHARMACOL, V25, P337
  • [6] KEATS AS, 1964, MOL MODIFICATION DRU, P170
  • [7] LARGENT BL, 1986, J PHARMACOL EXP THER, V238, P739
  • [8] PSYCHOTOMIMETIC OPIATE RECEPTORS LABELED AND VISUALIZED WITH (+)-[H-3]3-(3-HYDROXYPHENYL)-N-(1-PROPYL)PIPERIDINE
    LARGENT, BL
    GUNDLACH, AL
    SNYDER, SH
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (15): : 4983 - 4987
  • [9] MARTIN WR, 1976, J PHARMACOL EXP THER, V197, P517
  • [10] A PRACTICAL COMPUTER-BASED APPROACH TO THE ANALYSIS OF RADIOLIGAND BINDING EXPERIMENTS
    MCPHERSON, GA
    [J]. COMPUTER PROGRAMS IN BIOMEDICINE, 1983, 17 (1-2): : 107 - 114