MECHANISM OF ACTION OF DIGITALIS - IS THE NA,K-ATPASE THE PHARMACOLOGICAL RECEPTOR

被引:64
作者
SCHWARTZ, A
WHITMER, K
GRUPP, G
GRUPP, I
ADAMS, RJ
LEE, SW
机构
[1] UNIV CINCINNATI,COLL MED,DEPT PHARMACOL & CELL BIOPHYS,CINCINNATI,OH 45267
[2] UNIV CINCINNATI,COLL MED,DEPT PHYSIOL,CINCINNATI,OH 45267
关键词
D O I
10.1111/j.1749-6632.1982.tb25746.x
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:253 / 271
页数:19
相关论文
共 37 条
[1]   HIGH-AFFINITY OUABAIN BINDING-SITE AND LOW-DOSE POSITIVE INOTROPIC EFFECT IN RAT MYOCARDIUM [J].
ADAMS, RJ ;
SCHWARTZ, A ;
GRUPP, G ;
GRUPP, I ;
LEE, SW ;
WALLICK, ET ;
POWELL, T ;
TWIST, VW ;
GATHIRAM, P .
NATURE, 1982, 296 (5853) :167-169
[2]   LONG-TERM DIGITALIS THERAPY IMPROVES LEFT-VENTRICULAR FUNCTION IN HEART-FAILURE [J].
ARNOLD, SB ;
BYRD, RC ;
MEISTER, W ;
MELMON, K ;
CHEITLIN, MD ;
BRISTOW, JD ;
PARMLEY, WW ;
CHATTERJEE, K .
NEW ENGLAND JOURNAL OF MEDICINE, 1980, 303 (25) :1443-1448
[3]   CHANGES IN CELLULAR NA+, K+, AND CA2+ CONTENTS, MONO-VALENT CATION-TRANSPORT RATE, AND CONTRACTILE STATE DURING WASHOUT OF CARDIAC-GLYCOSIDES FROM CULTURED CHICK HEART-CELLS [J].
BARRY, WH ;
BIEDERT, S ;
MIURA, DS ;
SMITH, TW .
CIRCULATION RESEARCH, 1981, 49 (01) :141-149
[4]   CARDIAC GLYCOSIDE RECEPTOR, (NA+ + K+)-ATPASE ACTIVITY AND FORCE OF CONTRACTION IN RAT-HEART [J].
ERDMANN, E ;
PHILIPP, G ;
SCHOLZ, H .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (24) :3219-3229
[5]  
ERDMANN E, 1981, 3RD INT C NA K ATP S
[6]   ENDOGENOUS DIGITALIS-LIKE ACTIVITY IN MAMMALIAN BRAIN [J].
FISHMAN, MC .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1979, 76 (09) :4661-4663
[7]  
FOLCH J, 1957, J BIOL CHEM, V226, P497
[8]  
GODFRAIND T, 1981, ARCH INT PHARMACOD T, V250, P316
[9]  
GODFRAIND T, 1981, HDB EXPT PHARM, V56, P381
[10]   DIGITALIS RECEPTOR DESENSITIZATION IN RAT VENTRICLE - OUABAIN PRODUCES 2 INOTROPIC EFFECTS [J].
GRUPP, IL ;
GRUPP, G ;
SCHWARTZ, A .
LIFE SCIENCES, 1981, 29 (26) :2789-2794