DEFINITION OF 2 DISTINCT MECHANISMS OF ACTION OF ANTIESTROGENS ON HUMAN-BREAST CANCER CELL-PROLIFERATION USING HYDROXYTRIPHENYLETHYLENES WITH HIGH-AFFINITY FOR THE ESTROGEN-RECEPTOR

被引:58
作者
SUTHERLAND, RL [1 ]
WATTS, CKW [1 ]
RUENITZ, PC [1 ]
机构
[1] UNIV GEORGIA, COLL PHARM, ATHENS, GA 30602 USA
关键词
D O I
10.1016/0006-291X(86)90763-1
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:523 / 529
页数:7
相关论文
共 20 条
[1]   CALMODULIN AND THE CELL-CYCLE - INVOLVEMENT IN REGULATION OF CELL-CYCLE PROGRESSION [J].
CHAFOULEAS, JG ;
BOLTON, WE ;
HIDAKA, H ;
BOYD, AE ;
MEANS, AR .
CELL, 1982, 28 (01) :41-50
[2]  
COEZY E, 1982, CANCER RES, V42, P317
[3]  
Jordan VC, 1986, ESTROGEN ANTIESTROGE
[4]  
KATZENELLENBOGEN BS, 1981, J BIOL CHEM, V256, P2908
[5]   TAMOXIFEN IS A CALMODULIN ANTAGONIST IN THE ACTIVATION OF CAMP PHOSPHODIESTERASE [J].
LAM, HYP .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 118 (01) :27-32
[6]  
LIPPMAN M, 1976, CANCER RES, V36, P4595
[7]   EFFECTS OF THE ANTIOESTROGEN TAMOXIFEN ON THE CELL-CYCLE KINETICS OF THE HUMAN-BREAST CANCER CELL-LINE, MCF-7 [J].
LYKKESFELDT, AE ;
LARSEN, JK ;
CHRISTENSEN, IJ ;
BRIAND, P .
BRITISH JOURNAL OF CANCER, 1984, 49 (06) :717-722
[8]   CALMODULIN-STIMULATED PHOSPHORYLATION OF 17-BETA-ESTRADIOL RECEPTOR ON TYROSINE [J].
MIGLIACCIO, A ;
ROTONDI, A ;
AURICCHIO, F .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (19) :5921-5925
[9]  
MILLER MA, 1983, CANCER RES, V43, P3094
[10]   DIFFERENTIAL-EFFECTS OF TAMOXIFEN AND ANALOGS WITH NONBASIC SIDE-CHAINS ON CELL-PROLIFERATION INVITRO [J].
MURPHY, LC ;
SUTHERLAND, RL .
ENDOCRINOLOGY, 1985, 116 (03) :1071-1078