CHARACTERIZATION OF THROMBOXANE A2 PROSTAGLANDIN H-2 (TXA2/PGH2) RECEPTORS OF RAT PLATELETS AND THEIR INTERACTION WITH TXA2/PGH2 RECEPTOR ANTAGONISTS

被引:31
作者
HANASAKI, K [1 ]
ARITA, H [1 ]
机构
[1] SHIONOGI & CO LTD, SHIONOGI RES LAB, FUKUSHIMA KU, OSAKA 553, JAPAN
关键词
D O I
10.1016/0006-2952(88)90075-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3923 / 3929
页数:7
相关论文
共 37 条
[1]   LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].
ARMSTRONG, RA ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964
[2]   THROMBOXANES - NEW GROUP OF BIOLOGICALLY-ACTIVE COMPOUNDS DERIVED FROM PROSTAGLANDIN ENDOPEROXIDES [J].
HAMBERG, M ;
SVENSSON, J ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1975, 72 (08) :2994-2998
[3]   PROSTAGLANDIN-D2 INTERACTS AT THROMBOXANE RECEPTOR-SITES ON GUINEA-PIG PLATELETS [J].
HAMIDBLOOMFIELD, S ;
WHITTLE, BJR .
BRITISH JOURNAL OF PHARMACOLOGY, 1986, 88 (04) :931-936
[4]   BIPHASIC ACTION OF PHOSPHOLIPASE-A IN COLLAGEN-STIMULATED RAT PLATELETS [J].
HANASAKI, K ;
NAKANO, T ;
ARITA, H .
JOURNAL OF BIOCHEMISTRY, 1987, 102 (01) :5-8
[5]   2 PHASIC GENERATION OF THROMBOXANE A2 BY THE ACTION OF COLLAGEN ON RAT PLATELETS [J].
HANASAKI, K ;
NAKANO, T ;
ARITA, H .
THROMBOSIS RESEARCH, 1987, 46 (03) :425-436
[6]   SPECIFIC RECEPTORS FOR THROMBOXANE-A2 IN CULTURED VASCULAR SMOOTH-MUSCLE CELLS OF RAT AORTA [J].
HANASAKI, K ;
NAKANO, K ;
KASAI, H ;
ARITA, H ;
OHTANI, K ;
DOTEUCHI, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1988, 150 (03) :1170-1175
[7]   EVIDENCE THAT THE RAT IS NOT AN APPROPRIATE MODEL TO STUDY THE ROLE OF PROSTAGLANDINS IN NORMAL OR ABNORMAL PLATELET-AGGREGATION [J].
HUZOORAKBAR ;
ANWER, K .
THROMBOSIS RESEARCH, 1986, 41 (04) :555-566
[8]  
JONES RL, 1983, LEUKOTRIENE RES, V11, P351
[9]  
KATSURA M, 1983, ADV PROSTAG THROMB L, V11, P351
[10]   CHARACTERIZATION OF U46619 BINDING IN UNACTIVATED, INTACT HUMAN-PLATELETS AND DETERMINATION OF BINDING-SITE AFFINITIES OF 4 TXA2/PGH2 RECEPTOR ANTAGONISTS (13-APA, BM 13.177, ONO 3708 AND SQ 29,548) [J].
KATTELMAN, EJ ;
VENTON, DL ;
LEBRETON, GC .
THROMBOSIS RESEARCH, 1986, 41 (04) :471-481