ANALOG OF ENKEPHALIN HAVING PROLONGED OPIATE-LIKE EFFECTS INVIVO

被引：133

作者：

WALKER, JM

BERNTSON, GG

SANDMAN, CA

COY, DH

SCHALLY, AV

KASTIN, AJ

机构：

[1] OHIO STATE UNIV,DEPT PSYCHOL,COLUMBUS,OH 43210

[2] VET ADM HOSP,NEW ORLEANS,LA 70112

来源：

SCIENCE | 1977年 / 196卷 / 4285期

关键词：

D O I：

10.1126/science.190683

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：85 / 87

页数：3

共 28 条

[1]

AKIL H, 1976, OPIATES ENDOGENOUS O, P63

[2] ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT [J].

BELLUZZI, JD ;

GRANT, N ;

GARSKY, V ;

SARANTAKIS, D ;

WISE, CD ;

STEIN, L .

NATURE, 1976, 260 (5552) :625-626

[3] BIOSYNTHETIC ORIGIN AND RECEPTOR CONFORMATION OF METHIONINE ENKEPHALIN [J].

BRADBURY, AF ;

SMYTH, DG ;

SNELL, CR .

NATURE, 1976, 260 (5547) :165-166

[4] EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE [J].

BUSCHER, HH ;

HILL, RC ;

ROMER, D ;

CARDINAUX, F ;

CLOSSE, A ;

HAUSER, D ;

PLESS, J .

NATURE, 1976, 261 (5559) :423-425

[5] OPIATE RECEPTOR AFFINITIES AND BEHAVIORAL-EFFECTS OF ENKEPHALIN - STRUCTURE-ACTIVITY RELATIONSHIP OF 10 SYNTHETIC PEPTIDE ANALOGS [J].

CHANG, JK ;

FONG, BTW ;

PERT, A ;

PERT, CB .

LIFE SCIENCES, 1976, 18 (12) :1473-1481

[6] SYNTHESIS AND BIOLOGICAL PROPERTIES OF [D-ALA-6,DES-GLY-NH2-10]-LH-RH ETHYLAMIDE, A PEPTIDE WITH GREATLY ENHANCED LH-RELEASING AND FSH-RELEASING ACTIVITY [J].

COY, DH ;

COY, EJ ;

SCHALLY, AV ;

VILCHEZM.J ;

HIROTSU, Y ;

ARIMURA, A .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1974, 57 (02) :335-340

[7] SYNTHESIS AND OPIOID ACTIVITIES OF STEREOISOMERS AND OTHER D-AMINO-ACID ANALOGS OF METHIONINE-ENKEPHALIN [J].

COY, DH ;

KASTIN, AJ ;

SCHALLY, AV ;

MORIN, O ;

CARON, NG ;

LABRIE, F ;

WALKER, JM ;

FERTEL, R ;

BERNTSON, GG ;

SANDMAN, CA .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1976, 73 (03) :632-638

[8]

D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74

[9] LACK OF EFFECT OF NALOXONE ON PAIN PERCEPTION IN HUMANS [J].

ELSOBKY, A ;

DOSTROVSKY, JO ;

WALL, PD .

NATURE, 1976, 263 (5580) :783-784

[10]

GARBAYJAUREGUIL.C, 1976, BIOCHEM BIOPHYS RES, V71, P588

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