BIOCHEMICAL AND PHARMACOLOGICAL CHARACTERIZATION OF THE BINDING OF THE SELECTIVE PEPTIDE-LEUKOTRIENE ANTAGONIST, H-3-ICI 198,615, TO LEUKOTRIENE-D4 RECEPTORS IN GUINEA-PIG LUNG MEMBRANES

被引:22
作者
AHARONY, D
FALCONE, RC
YEE, YK
HESP, B
GILES, RE
KRELL, RD
机构
关键词
D O I
10.1111/j.1749-6632.1988.tb38539.x
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:162 / 180
页数:19
相关论文
共 33 条
[1]   DISCRIMINATIVE EFFECT OF GAMMA-GLUTAMYL-TRANSFERASE TRANSPEPTIDASE INHIBITORS ON METABOLISM OF LEUKOTRIENE-C4 IN PERITONEAL-CELLS [J].
AHARONY, D ;
DOBSON, P .
LIFE SCIENCES, 1984, 35 (21) :2135-2142
[2]  
AHARONY D, 1987, J PHARMACOL EXP THER, V243, P921
[3]   SELECTIVE INHIBITOR OF SLOW REACTING SUBSTANCE OF ANAPHYLAXIS [J].
AUGSTEIN, J ;
FARMER, JB ;
LEE, TB ;
SHEARD, P ;
TATTERSALL, ML .
NATURE-NEW BIOLOGY, 1973, 245 (146) :215-217
[4]  
BUCKNER CK, 1986, J PHARMACOL EXP THER, V237, P558
[5]   EVIDENCE FOR A SIMILAR RECEPTOR-SITE FOR BINDING OF [H-3] LEUKOTRIENE-E4 AND [H-3] LEUKOTRIENE-D4 TO THE GUINEA-PIG CRUDE LUNG MEMBRANE [J].
CHENG, JB ;
TOWNLEY, RG .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 122 (03) :949-954
[6]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[7]   EFFECTS OF LEUKOTRIENES-C4 AND LEUKOTRIENE-D4 ON GLYCOPROTEIN AND LYSOZYME SECRETION BY HUMAN BRONCHIAL-MUCOSA [J].
COLES, SJ ;
NEILL, KH ;
REID, LM ;
AUSTEN, KF ;
NII, Y ;
COREY, EJ ;
LEWIS, RA .
PROSTAGLANDINS, 1983, 25 (02) :155-170
[8]  
DELEAN A, 1980, J BIOL CHEM, V255, P7108
[9]   COMPARATIVE AIRWAY AND VASCULAR ACTIVITIES OF LEUKOTRIENE-C-1 AND LEUKOTRIENE-D INVIVO AND INVITRO [J].
DRAZEN, JM ;
AUSTEN, KF ;
LEWIS, RA ;
CLARK, DA ;
GOTO, G ;
MARFAT, A ;
COREY, EJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (07) :4354-4358
[10]   EVIDENCE FOR MULTIPLE LEUKOTRIENE-D4 RECEPTORS IN SMOOTH-MUSCLE [J].
FLEISCH, JH ;
RINKEMA, LE ;
BAKER, SR .
LIFE SCIENCES, 1982, 31 (06) :577-581