REACTIONS OF 3-(TETRAHYDROPYRID-4-YL)-INDOLES WITH DIENOPHILES - NEW HETEROCYCLIC FUNCTIONALIZED INDOLES AND PYRIDO[C]ANNELLATED CARBAZOLES

被引：9

作者：

MEDIOSIMON, M

OTTO, C

PINDUR, U

机构：

[1] UNIV VALENCIA,FAC PHARM,DEPT ORGAN CHEM,VALENCIA,SPAIN

[2] UNIV MAINZ,FACHBEREICH CHEM & PHARM,INST PHARM,W-6500 MAINZ 1,GERMANY

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 15期

关键词：

D O I：

10.1016/S0040-4039(00)74326-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

First reactions of 3-(1,2,3,6-tetrahydropyrid-4-yl)-indoles 1 with a variety of carbo- and heterodienophiles are described. These reactions provide a new access to heterocyclic functionalized indoles and pyrido[c]annellated carbazoles, compounds of interest as potential antidepressive and antitumor active agents.

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页码：1771 / 1774

页数：4

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