DEVELOPMENT OF GLUCOCORTICOID ANTAGONISTS

被引:27
作者
CHROUSOS, GP
CUTLER, GB
SAUER, M
SIMONS, SS
LORIAUX, DL
机构
[1] NIADDKD,CHEM LAB,BETHESDA,MD 20205
[2] GEORGE WASHINGTON UNIV,DEPT PHARMACOL,WASHINGTON,DC 20006
关键词
D O I
10.1016/0163-7258(83)90041-4
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:263 / 281
页数:19
相关论文
共 39 条
[1]  
ACS Z, 1975, EXPERIENTIA, V31, P1365
[2]  
AXELROD JR, 1954, ENDOCRINOLOGY, V55, P568
[3]   DELTA-1,9(11)-11-DEOXYCORTISOL - AN IMPROVED GLUCOCORTICOID ANTAGONIST [J].
CHROUSOS, GP ;
BARNES, KM ;
SAUER, MA ;
LORIAUX, DL ;
CUTLER, GB .
ENDOCRINOLOGY, 1980, 107 (02) :472-477
[4]   DELTA-1-11-OKA-11-DEOXYCORTISOL - A NEW ANTIGLUCOCORTICOID WITH ACTIVITY INVIVO [J].
CHROUSOS, GP ;
SAUER, MA ;
LORIAUX, DL ;
CUTLER, GB .
STEROIDS, 1982, 40 (04) :425-431
[5]   ESTROGEN RECEPTOR - ANTIESTROGEN COMPLEX - ATYPICAL BINDING BY UTERINE NUCLEI AND EFFECTS ON UTERINE GROWTH [J].
CLARK, JH ;
ANDERSON, JN ;
PECK, EJ .
STEROIDS, 1973, 22 (05) :707-718
[6]  
Clark JH, 1982, PHARMACOL THERAPEUT, V15, P467
[7]   11-DEOXYCORTISOL - GLUCOCORTICOID ANTAGONIST INVIVO [J].
CUTLER, GB ;
BARNES, KM ;
SAUER, MA ;
LORIAUX, DL .
ENDOCRINOLOGY, 1979, 104 (06) :1839-1844
[8]  
DELEAN A, 1978, MOL PHARM, V15, P60
[9]   GLUCOCORTICOID ACTIVITY OF VARIOUS PROGESTERONE ANALOGS - CORRELATION BETWEEN SPECIFIC BINDING IN THYMUS AND LIVER AND BIOLOGIC ACTIVITY [J].
DISORBO, D ;
ROSEN, F ;
MCPARTLAND, RP ;
MILHOLLAND, RJ .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1977, 286 (MAR11) :355-368
[10]  
DORFMAN RI, 1964, METHODS HORMONE RES, V2, P325