INHIBITION OF HISTAMINE SYNTHESIS INVITRO AND INVIVO BY S-ALPHA-FLUOROMETHYLHISTIDINE

被引:43
作者
DUGGAN, DE [1 ]
HOOKE, KF [1 ]
MAYCOCK, AL [1 ]
机构
[1] MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065
关键词
D O I
10.1016/0006-2952(84)90013-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:4003 / 4009
页数:7
相关论文
共 17 条
[1]  
BARTHOLEYNS J, 1982, CONTRACEPTION, V26, P535, DOI 10.1016/0010-7824(82)90152-4
[2]  
BEAVEN M, 1978, MONOGRAPHS ALLERGY, V13
[3]  
BEAVEN MA, 1968, J PHARMACOL EXP THER, V161, P320
[4]   MODIFICATION OF ENZYMATIC ISOTOPIC ASSAY OF HISTAMINE AND ITS APPLICATION TO MEASUREMENT OF HISTAMINE IN TISSUES, SERUM AND URINE [J].
BEAVEN, MA ;
HORAKOVA, Z ;
JACOBSEN, S .
CLINICA CHIMICA ACTA, 1972, 37 (NMAR) :91-+
[5]   HISTAMINE TURNOVER IN RAT-BRAIN [J].
DISMUKES, K ;
SNYDER, SH .
BRAIN RESEARCH, 1974, 78 (03) :467-481
[6]  
DUGGAN D, 1981, PHARMACOLOGIST, V23, P161
[7]   IMMUNOCHEMICAL CROSS-REACTIVITY OF THE ANTIBODY ELICITED AGAINST L-HISTIDINE DECARBOXYLASE PURIFIED FROM THE WHOLE BODIES OF FETAL RATS WITH THE ENZYME FROM RAT-BRAIN [J].
FUKUI, H ;
WATANABE, T ;
WADA, H .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1980, 93 (01) :333-339
[8]   INHIBITION OF HISTAMINE SYNTHESIS IN BRAIN BY ALPHA-FLUOROMETHYLHISTIDINE, A NEW IRREVERSIBLE INHIBITOR - INVITRO AND INVIVO STUDIES [J].
GARBARG, M ;
BARBIN, G ;
RODERGAS, E ;
SCHWARTZ, JC .
JOURNAL OF NEUROCHEMISTRY, 1980, 35 (05) :1045-1052
[9]   HISTIDINE DECARBOXLASE IN FETAL RAT [J].
HAKANSON, R .
BIOCHEMICAL PHARMACOLOGY, 1963, 12 (11) :1289-&
[10]   SELECTIVE INHIBITORS OF BIOSYNTHESIS OF AMINERGIC NEUROTRANSMITTERS [J].
KOLLONITSCH, J ;
PATCHETT, AA ;
MARBURG, S ;
MAYCOCK, AL ;
PERKINS, LM ;
DOLDOURAS, GA ;
DUGGAN, DE ;
ASTER, SD .
NATURE, 1978, 274 (5674) :906-908