NG-2,2,5,7,8-PENTAMETHYLCHROMAN-6-SULFONYL-L-ARGININE - A NEW ACID LABILE DERIVATIVE FOR PEPTIDE-SYNTHESIS

被引：97

作者：

RAMAGE, R

GREEN, J

机构：

来源：

TETRAHEDRON LETTERS | 1987年 / 28卷 / 20期

关键词：

D O I：

10.1016/S0040-4039(00)96103-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：2287 / 2290

页数：4

共 18 条

[1] SIDE-CHAIN PROTECTED N-ALPHA-FLUORENYLMETHOXYCARBONYLAMINO-ACIDS FOR SOLID-PHASE PEPTIDE-SYNTHESIS - N-ALPHA-FLUORENYLMETHOXYCARBONYL-NG-4-METHOXY-2,3,6-TRIMETHYLBENZENESULPHONYL-L-ARGININE [J].

ATHERTON, E ;

SHEPPARD, RC ;

WADE, JD .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1983, (19) :1060-1062

[2] SYNTHESE DE LA L-HISTIDYL-L-PHENYLALANYL-L-ARGINYL-L-TRYPTOPHANYL-GLYCYL-EPSILON-CBO-L-LYSYL-L-PROLYL-L-VALYLAMIDE [J].

BOISSONNAS, RA ;

GUTTMANN, S ;

HUGUENIN, RL ;

JAQUENOUD, PA ;

SANDRIN, E .

HELVETICA CHIMICA ACTA, 1958, 41 (06) :1867-1882

[3]

FUJINO M, 1981, CHEM PHARM BULL, V29, P2825

[4] 4-METHOXY-2,6-DIMETHYLBENZENESULPHONYL (MDS) - A NEW PROTECTING GROUP OF THE GUANIDINO FUNCTION IN PEPTIDE-SYNTHESIS [J].

FUJINO, M ;

NISHIMURA, O ;

WAKIMASU, M ;

KITADA, C .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1980, (14) :668-669

[5]

JACKSON AG, 1976, TETRAHEDRON LETT, P3627

[6] EFFICIENT DEPROTECTION OF NG-TOSYLARGININE WITH A THIOANISOLE-TRIFLUOROMETHANESULPHONIC ACID SYSTEM [J].

KISO, Y ;

SATOMI, M ;

UKAWA, K ;

AKITA, T .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1980, (22) :1063-1064

[7] EFFICIENT REMOVAL OF N-BENZYLOXYCARBONYL GROUP BY A PUSH-PULL MECHANISM USING THIOANISOLE-TRIFLUOROACETIC ACID, EXEMPLIFIED BY A SYNTHESIS OF MET-ENKEPHALIN [J].

KISO, Y ;

UKAWA, K ;

AKITA, T .

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1980, (03) :101-102

[8] IMPROVED SYNTHESIS OF BRADYKININ [J].

MAZUR, RH ;

PLUME, G .

EXPERIENTIA, 1968, 24 (07) :661-&

[9]

NISHIMURA O, 1976, CHEM PHARM BULL, V24, P1568

[10] SOME NEW ARENESULFONATE LEAVING GROUPS LESS REACTIVE THAN P-TOLUENESULFONATE GROUP [J].

PALEOS, CM ;

VARVERI, FS ;

GREGORIO.GA .

JOURNAL OF ORGANIC CHEMISTRY, 1974, 39 (24) :3594-3595

← 1 2 →