ANTIINFLAMMATORY AGENTS .3. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF 2-AMINO-3-BENZOYLPHENYLACETIC ACID AND ANALOGS

被引：57

作者：

WALSH, DA

MORAN, HW

SHAMBLEE, DA

UWAYDAH, IM

WELSTEAD, WJ

SANCILIO, LF

DANNENBURG, WN

机构：

[1] AH ROBINS CO, DEPT PHARMACOL, RICHMOND, VA 23261 USA

[2] AH ROBINS CO, DEPT MOLEC BIOL, RICHMOND, VA 23261 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1984年 / 27卷 / 11期

关键词：

D O I：

10.1021/jm00377a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1379 / 1388

页数：10

共 18 条

[1] CONFORMATIONAL REQUIREMENTS AT THE PROSTAGLANDIN CYCLOOXYGENASE RECEPTOR-SITE - TEMPLATE FOR DESIGNING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS [J].

APPLETON, RA ;

BROWN, K .

PROSTAGLANDINS, 1979, 18 (01) :29-34

[2]

BAYS DE, 1974, Patent No. 3828093

[3]

BEKEMEIER H, 1982, TRENDS INFLAMMATIO S, V10, P17

[4] USE OF HALOGEN-SULFIDE COMPLEXES IN SYNTHESIS OF INDOLES, OXINDOLES, AND ALKYLATED AROMATIC-AMINES [J].

GASSMAN, PG ;

VANBERGE.TJ ;

GRUETZMA.G .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1973, 95 (19) :6508-6509

[5]

GASSMAN PG, 1974, J AM CHEM SOC, V96, P5508, DOI 10.1021/ja00824a029

[6]

GASSMAN PG, 1975, 169TH NAT M AM CHEM

[7] SYNTHESIS OF 2-AMINO-3-BENZOYLPHENYLACETIC ACID [J].

LO, YS ;

WALSH, DA ;

WELSTEAD, WJ ;

MAYS, RP ;

ROSE, EK ;

CAUSEY, DH ;

DUNCAN, RL .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1980, 17 (08) :1663-1664

[8]

MONTAGNE PJ, 1916, CHEM BER, V49, P2262

[9] APPLICATION OF SEQUENTIAL-ANALYSIS TO EVANS BLUE-CARRAGEENAN-INDUCED PLEURAL EFFUSION FOR SCREENING COMPOUNDS FOR ANTIINFLAMMATORY ACTIVITY [J].

SANCILIO, LF ;

FISHMAN, A .

TOXICOLOGY AND APPLIED PHARMACOLOGY, 1973, 26 (04) :575-584

[10] AHR-5850 - POTENT ANTI-INFLAMMATORY COMPOUND [J].

SANCILIO, LF ;

REESE, DL ;

CHEUNG, S ;

ALPHIN, RS .

AGENTS AND ACTIONS, 1977, 7 (01) :133-144

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